SCHEMBL7569727

SCHEMBL7569727

CCOc1cc2c(cc1OC)C(=[C]C#N)N[C@@H](C)C2

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ACHE P22303 2/20 0.44
HTR2A P28223 2/20 0.40
HTR2C P28335 2/20 0.40
HTR2B P41595 2/20 0.40
HTR1A P08908 1/20 0.40
HTR7 P34969 1/20 0.40
PDE4D Q08499 4/20 0.38
PDE4A P27815 4/20 0.38
PDE4B Q07343 2/20 0.38
PDE4C Q08493 2/20 0.38
KDM4E B2RXH2 2/20 0.36
ALDH1A1 P00352 1/20 0.36
KMT2A Q03164 1/20 0.36
MAPK1 P28482 1/20 0.34
CASP1 P29466 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7425283 0.79 ACHE (0.42) ACHEHTR2AHTR2CHTR2BHTR1A
Bromide SCHEMBL7430276 0.72 ACHE (0.36) ACHEHTR2AHTR2CHTR2BHTR1A
SCHEMBL3370335 0.69 ALDH1A1 (0.56) ACHEKDM4EALDH1A1KMT2AMAPK1
SCHEMBL3370337 0.69 ALDH1A1 (0.56) ACHEKDM4EALDH1A1KMT2AMAPK1
SCHEMBL3367902 0.65 KDM4E (0.63) ACHEKDM4EALDH1A1KMT2A
SCHEMBL3367895 0.65 KDM4E (0.63) ACHEKDM4EALDH1A1KMT2A
SCHEMBL22029967 0.64 MAPT (0.70) ACHEHTR2AHTR2CHTR2BHTR1A
SCHEMBL23369357 0.63 PDE4A (0.56) ACHEHTR2AHTR2CHTR2BHTR1A
SCHEMBL28662301 0.62 KDM4E (0.57) HTR2AHTR2CHTR2BPDE4DPDE4A
SCHEMBL28311309 0.62 KDM4E (0.57) HTR2AHTR2CHTR2BPDE4DPDE4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001064647-A1 ISOQUINOLINE DERIVATIVES AS PDE4 INHIBITORS SANOFI-SYNTHELABO (FR) 2001-09-07 WO disclosed