SCHEMBL7570328

SCHEMBL7570328

O=C1N=C(O)C(c2ccc(C(F)(F)F)cc2)=NC1Cc1ccc(-c2ccccc2)cc1

nearest known ligand 0.45

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CES2 O00748 2/20 0.45
KIF11 P52732 1/20 0.42
CCKAR P32238 3/20 0.39
CCKBR P32239 3/20 0.39
NPSR1 Q6W5P4 1/20 0.38
BACE1 P56817 1/20 0.38
GLO1 Q04760 1/20 0.38
LMNA P02545 1/20 0.36
HTT P42858 1/20 0.36
FFAR1 O14842 1/20 0.36
HDAC3 O15379 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
ACLY P53396 1/20 0.36
EPHX2 P34913 1/20 0.36
CCNC P24863 1/20 0.35
CDK8 P49336 1/20 0.35
SLC13A5 Q86YT5 1/20 0.35
PTPN1 P18031 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7572646 0.88 BDKRB2 (0.41) CES2LMNAHTTHDAC3HDAC6
SCHEMBL7572631 0.87 CES2 (0.42) CES2CCKARCCKBRHDAC3HDAC6
SCHEMBL7572458 0.85 BDKRB2 (0.42) CES2HDAC3HDAC6
SCHEMBL7572718 0.84 CES2 (0.43) CES2LMNAHDAC3HDAC6
SCHEMBL7571711 0.82 CES2 (0.38) CES2CCKARCCKBRLMNAHDAC3
SCHEMBL7571381 0.81 HDAC3 (0.42) CCKARCCKBRHDAC3HDAC6
SCHEMBL7575515 0.80 ESR1 (0.37) BACE1LMNAHDAC3HDAC6
SCHEMBL7571208 0.79 NPC1 (0.44) CES2NPSR1HDAC3HDAC6
SCHEMBL7576544 0.79 CES2 (0.44) CES2LMNAHDAC3HDAC6
SCHEMBL7571399 0.79 PTPN5 (0.38) CCKBRHTTHDAC3HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002085369-A1 INHIBITORS OF ANTHRAX LETHAL FACTOR ACTIVITY STRUCTURAL BIOINFORMATICS, INC. (US) 2002-10-31 WO disclosed