SCHEMBL7576544

SCHEMBL7576544

Cc1ccc(C2=NC(Cc3ccccc3)C(=O)N=C2O)cc1

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CES2 O00748 5/20 0.44
KLK7 P49862 1/20 0.40
MAPT P10636 2/20 0.39
LMNA P02545 1/20 0.39
BDKRB2 P30411 2/20 0.37
HDAC3 O15379 2/20 0.37
HDAC6 Q9UBN7 2/20 0.37
HDAC1 Q13547 1/20 0.37
HDAC8 Q9BY41 1/20 0.37
ALOX5 P09917 1/20 0.36
BRD4 O60885 2/20 0.35
KDM4E B2RXH2 1/20 0.35
BRD2 P25440 1/20 0.35
BRD3 Q15059 1/20 0.35
MEN1 O00255 1/20 0.34
ALDH1A1 P00352 1/20 0.34
KMT2A Q03164 1/20 0.34
RGS4 P49798 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7572718 0.95 CES2 (0.43) CES2KLK7MAPTLMNABDKRB2
SCHEMBL7572646 0.91 BDKRB2 (0.41) CES2LMNABDKRB2HDAC3HDAC6
SCHEMBL7572458 0.90 BDKRB2 (0.42) CES2BDKRB2HDAC3HDAC6HDAC1
SCHEMBL7571381 0.89 HDAC3 (0.42) BDKRB2HDAC3HDAC6HDAC1HDAC8
SCHEMBL7571711 0.87 CES2 (0.38) CES2LMNABDKRB2HDAC3HDAC6
SCHEMBL7571208 0.87 NPC1 (0.44) CES2MAPTBDKRB2HDAC3HDAC6
SCHEMBL7575808 0.84 CES2 (0.41) CES2LMNABDKRB2HDAC3HDAC6
SCHEMBL7576399 0.83 CNR2 (0.35) CES2BDKRB2HDAC3HDAC6HDAC1
SCHEMBL7576579 0.83 RARB (0.44) MAPTLMNABDKRB2KDM4EMEN1
SCHEMBL7572631 0.82 CES2 (0.42) CES2BDKRB2HDAC3HDAC6HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002085369-A1 INHIBITORS OF ANTHRAX LETHAL FACTOR ACTIVITY STRUCTURAL BIOINFORMATICS, INC. (US) 2002-10-31 WO disclosed