SCHEMBL757064

SCHEMBL757064

Nc1ccccc1CCc1cc(CCc2ccccc2)ncn1

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 1/20 0.43
BACE1 P56817 2/20 0.42
KCNH2 Q12809 1/20 0.42
NOS1 P29475 1/20 0.41
ADK P55263 1/20 0.41
MAOA P21397 4/20 0.41
MAOB P27338 4/20 0.41
HTR1A P08908 2/20 0.40
DRD2 P14416 2/20 0.40
ABCB1 P08183 2/20 0.40
DHFR P00374 1/20 0.40
OPRL1 P41146 1/20 0.39
EGFR P00533 1/20 0.38
ATP4A P20648 1/20 0.38
ATP4B P51164 1/20 0.38
KDM4E B2RXH2 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13754947 0.84 KCNH2 (0.56) BACE1KCNH2NOS1MAOAMAOB
SCHEMBL88596 0.82 MAOB (0.56) SIGMAR1MAOAMAOBHTR1ADRD2
Hydrochloric Acid SCHEMBL8746158 0.80 MAOB (0.58) SIGMAR1MAOAMAOBHTR1ADRD2
SCHEMBL6810696 0.80 HTR2A (0.54) BACE1KCNH2NOS1MAOAMAOB
SCHEMBL752310 0.76 TDP1 (0.54) BACE1KCNH2NOS1EGFRKDM4E
SCHEMBL13754981 0.76 KCNH2 (0.47) BACE1KCNH2NOS1MAOAMAOB
SCHEMBL27756279 0.76 KCNH2 (0.47) BACE1KCNH2NOS1MAOAMAOB
SCHEMBL2486170 0.73 EPHX1 (0.53) SIGMAR1BACE1KCNH2NOS1MAOA
SCHEMBL752939 0.73 KCNH2 (0.47) BACE1KCNH2NOS1MAOBEGFR
SCHEMBL3432650 0.72 MAP2K7 (0.44) KCNH2EGFRKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20170066754-A1 ANTIVIRAL AGENT SHIONOGI & CO., LTD. (JP) 2017-03-09 US disclosed
US-9572813-B2 Antiviral agent SHIONOGI & CO., LTD. (JP) 2017-02-21 US disclosed
US-20150202208-A1 ANTIVIRAL AGENT SHIONOGI & CO., LTD. (JP) 2015-07-23 US disclosed
EP-1422218-B1 ANTIVIRAL AGENT SHIONOGI & CO (JP) 2012-03-21 EP disclosed
EP-2181985-B1 Antiviral Agent SHIONOGI & CO (JP) 2011-10-26 EP disclosed
US-20040229909-A1 Antiviral agent SHIONOGI & CO., LTD. (JP) 2004-11-18 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040229909-A1 Antiviral agent ZC3HAV1, ZC3HAV1L, DUT SIGMAR1 1836/4885BACE1 1504/4885KCNH2 3468/4885
US-20150202208-A1 ANTIVIRAL AGENT ZC3HAV1, ZC3HAV1L, CCNI SIGMAR1 1890/4885BACE1 1681/4885KCNH2 3830/4885
US-20170066754-A1 ANTIVIRAL AGENT ZC3HAV1, ZC3HAV1L, CCNI SIGMAR1 1890/4885BACE1 1681/4885KCNH2 3830/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.