SCHEMBL7570871

SCHEMBL7570871

CC(C)(C)n1nc(CCc2ccc(Cl)cc2)nc1CCO

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.36
CYP3A4 P08684 1/20 0.36
KMT2A Q03164 2/20 0.33
NPC1 O15118 2/20 0.33
RAB9A P51151 2/20 0.33
PDE4B Q07343 2/20 0.33
MEN1 O00255 1/20 0.33
TSHR P16473 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
CYP11B1 P15538 1/20 0.32
CYP11B2 P19099 1/20 0.32
P2RX3 P56373 1/20 0.32
TAAR1 Q96RJ0 1/20 0.32
SLC6A2 P23975 1/20 0.32
HTR2A P28223 1/20 0.32
SLC6A4 P31645 1/20 0.32
HRH1 P35367 1/20 0.32
HTR2B P41595 1/20 0.32
CHRNA4 P43681 1/20 0.32
SLC6A3 Q01959 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4978016 0.72 ALDH1A1 (0.41) ALDH1A1CYP3A4KMT2ANPC1RAB9A
SCHEMBL4978019 0.67 ALDH1A1 (0.38) ALDH1A1CYP3A4KMT2ANPC1RAB9A
SCHEMBL77492 0.66 CA2 (0.59) ALDH1A1TSHRTAAR1
Alcohol SCHEMBL5328957 0.65 CA2 (0.52) ALDH1A1TAAR1
SCHEMBL28309115 0.62 CA2 (0.54) ALDH1A1TSHRTAAR1
SCHEMBL8439467 0.62 ALDH1A1 (0.36) ALDH1A1CYP3A4KMT2AMEN1SLC6A4
SCHEMBL2135113 0.61 TAAR1 (0.68) TAAR1SLC6A4
SCHEMBL10789850 0.61 CA2 (0.52) KMT2AMEN1TAAR1
SCHEMBL11000396 0.61 MAOB (0.59) ALDH1A1TAAR1
SCHEMBL16663705 0.60 TAAR1 (0.54) TSHRTAAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 17 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002074084-A1 NEORUSTMICIN D DERIVATIVES AS FUNGICIDES BASF AKTIENGESELLSCHAFT (DE) 2002-09-26 WO disclosed
EP-1037893-A1 USE OF NITROETHANE DERIVATIVES AS MICROBICIDES AND SPECIFIC NITROETHANE DERIVATIVES BASF AKTIENGESELLSCHAFT (DE) 2000-09-27 EP disclosed
US-6114342-A 2-(O-[pyrimidin-4-yl]methylenoxy)phenylacetic acid derivatives and their use for controlling harmful fungi and animal pests BASF AKTIENGESELLSCHAFT (DE) 2000-09-05 US disclosed
EP-1017671-A1 NOVEL BENZAMIDOXIM DERIVATIVES, INTERMEDIATE PRODUCTS AND METHODS FOR PREPARING THEM, AND THEIR USE AS FUNGICIDES BASF AKTIENGESELLSCHAFT (DE) 2000-07-12 EP disclosed
EP-1003725-A1 FLUOROPYRAZOLE-BIPHENYLAMIDE FUNGICIDES BASF AKTIENGESELLSCHAFT (DE) 2000-05-31 EP disclosed
WO-1999031108-A1 USE OF NITROETHANE DERIVATIVES AS MICROBICIDES AND SPECIFIC NITROETHANE DERIVATIVES BASF AKTIENGESELLSCHAFT (DE) 1999-06-24 WO disclosed
WO-1999029671-A1 3-PYRAZOLE-1-YL BENZOIC ACID DERIVATIVES BASF AKTIENGESELLSCHAFT (DE) 1999-06-17 WO disclosed
EP-0906271-A1 CARBAMOYL CARBOXYLIC ACID AMIDE OXIMES BASF AKTIENGESELLSCHAFT (DE) 1999-04-07 EP disclosed
WO-1999014188-A1 NOVEL BENZAMIDOXIM DERIVATIVES, INTERMEDIATE PRODUCTS AND METHODS FOR PREPARING THEM, AND THEIR USE AS FUNGICIDES BASF AKTIENGESELLSCHAFT (DE) 1999-03-25 WO disclosed
WO-1999009013-A1 FLUOROPYRAZOLE-BIPHENYLAMIDE FUNGICIDES BASF AKTIENGESELLSCHAFT (DE) 1999-02-25 WO disclosed
EP-0852579-A1 FUNGICIDAL QUINOLINES BASF AKTIENGESELLSCHAFT (DE) 1998-07-15 EP disclosed
WO-1997046518-A1 CARBAMOYL CARBOXYLIC ACID AMIDE OXIMES BASF AKTIENGESELLSCHAFT (DE) 1997-12-11 WO disclosed
EP-0778824-A1 CARBAMOYL CARBOXYLIC ACID AMIDES BASF AKTIENGESELLSCHAFT (DE) 1997-06-18 EP disclosed
WO-1997010215-A1 FUNGICIDAL QUINOLINES BASF AKTIENGESELLSCHAFT (DE) 1997-03-20 WO disclosed
WO-1996007638-A1 CARBAMOYL CARBOXYLIC ACID AMIDES BASF AKTIENGESELLSCHAFT (DE) 1996-03-14 WO disclosed
WO-1995023785-A1 CARBAMOYL CARBOXYLIC ACID AMIDES, PROCESS FOR PRODUCING THEM AND THEIR USE AS FUNGICIDES BASF AKTIENGESELLSCHAFT (DE) 1995-09-08 WO disclosed
WO-1995023784-A1 CARBAMOYL CARBOXYLIC ACID AMIDES, PROCESS FOR PRODUCING THEM AND THEIR USE AS FUNGICIDES BASF AKTIENGESELLSCHAFT (DE) 1995-09-08 WO disclosed