SCHEMBL7571578

SCHEMBL7571578

COC(=O)c1ccc(NS(=O)(=O)C(F)(F)F)c(NS(=O)(=O)c2cc(Cl)sc2Cl)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.48
ACLY P53396 5/20 0.47
CDK1 P06493 1/20 0.43
CCNB1 P14635 1/20 0.43
CCNA2 P20248 1/20 0.43
CCND1 P24385 1/20 0.43
CDK2 P24941 1/20 0.43
CDK7 P50613 1/20 0.43
CCNH P51946 1/20 0.43
CCNA1 P78396 1/20 0.43
CDK6 Q00534 1/20 0.43
S100A9 P06702 3/20 0.42
CMA1 P23946 4/20 0.41
PDK1 Q15118 2/20 0.41
PDK2 Q15119 2/20 0.41
PDK3 Q15120 2/20 0.41
PDK4 Q16654 2/20 0.41
CYP2C9 P11712 2/20 0.41
PFKFB3 Q16875 1/20 0.40
MCL1 Q07820 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7569703 0.81 ACLY (0.52) TDP1ACLYCDK1CCNB1CCNA2
SCHEMBL7572367 0.74 SMN1; SMN2 (0.50) ACLYCMA1CYP2C9
SCHEMBL7149263 0.71 MAPT (0.58) TDP1ACLY
SCHEMBL7573034 0.70 ACLY (0.53) ACLYCMA1CYP2C9PFKFB3
SCHEMBL15830513 0.70 CYP2C9 (0.64) ACLYCYP2C9
SCHEMBL7593518 0.70 ACLY (0.61) TDP1ACLYCDK1CCNB1CCNA2
SCHEMBL7572555 0.69 CYP2C9 (0.60) ACLYCYP2C9
SCHEMBL7589604 0.69 S100A9 (0.51) TDP1ACLYCDK1CCNB1CCNA2
SCHEMBL7592196 0.69 CDK1 (0.63) TDP1ACLYCDK1CCNB1CCNA2
SCHEMBL15830515 0.69 ALDH1A1 (0.62) CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1239852-A2 BISSULFONAMIDE DERIVATIVES AS ENZYME INHIBITORS Arrow Therapeutics Limited (GB) 2002-09-18 EP disclosed
WO-2001028537-A2 BISSULFONAMIDE DERIVATIVES AS ENZYME INHIBITORS ARROW THERAPEUTICS LIMITED (GB) 2001-04-26 WO disclosed