SCHEMBL7573034

SCHEMBL7573034

COC(=O)c1ccc(NS(=O)(=O)c2cccc(Cl)c2C)c(NS(=O)(=O)c2cccc(Cl)c2C)c1

nearest known ligand 0.53

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ACLY P53396 2/20 0.53
CYP2C9 P11712 3/20 0.48
SLC40A1 Q9NP59 1/20 0.48
PFKFB3 Q16875 1/20 0.47
PFKFB4 Q16877 1/20 0.47
HSD11B1 P28845 2/20 0.47
ALDH1A1 P00352 4/20 0.46
MAPT P10636 2/20 0.46
TSHR P16473 2/20 0.46
NPSR1 Q6W5P4 1/20 0.46
CMA1 P23946 3/20 0.46
KDM4E B2RXH2 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
TP53 P04637 1/20 0.46
CCR4 P51679 1/20 0.46
EDNRB P24530 1/20 0.45
EDNRA P25101 1/20 0.45
POLB P06746 1/20 0.45
IDH1 O75874 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7572428 0.90 ALDH1A1 (0.54) SLC40A1HSD11B1ALDH1A1MAPTTSHR
SCHEMBL3873411 0.81 PFKFB3 (0.48) CYP2C9PFKFB3PFKFB4HSD11B1ALDH1A1
SCHEMBL7588152 0.79 SLC40A1 (0.59) SLC40A1HSD11B1ALDH1A1MAPTTSHR
SCHEMBL7594250 0.78 SLC40A1 (0.66) SLC40A1HSD11B1ALDH1A1CCR4EDNRB
SCHEMBL7594652 0.78 SLC40A1 (0.53) ACLYSLC40A1HSD11B1EDNRBEDNRA
SCHEMBL12406979 0.77 KDM4E (0.60) ACLYCYP2C9SLC40A1PFKFB3PFKFB4
SCHEMBL3873274 0.76 FABP4 (0.49) PFKFB3PFKFB4ALDH1A1MAPTTP53
SCHEMBL7578810 0.76 SLC40A1 (0.64) SLC40A1HSD11B1CCR4EDNRBEDNRA
SCHEMBL7591197 0.76 PTGES2 (0.59) ACLYSLC40A1HSD11B1CCR4EDNRB
SCHEMBL2174600 0.76 FFAR4 (0.61) CYP2C9ALDH1A1MAPTTSHRNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1239852-A2 BISSULFONAMIDE DERIVATIVES AS ENZYME INHIBITORS Arrow Therapeutics Limited (GB) 2002-09-18 EP disclosed
WO-2001028537-A2 BISSULFONAMIDE DERIVATIVES AS ENZYME INHIBITORS ARROW THERAPEUTICS LIMITED (GB) 2001-04-26 WO disclosed