SCHEMBL7573077

SCHEMBL7573077

CS(=O)(=O)Oc1ccc(C2=C(Cc3ccc(OCCN4CCCC4)cc3)c3ccc(O)cc3C2)cc1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 19/20 0.60
ESR2 Q92731 15/20 0.60
MLNR O43193 1/20 0.45
ABCB11 O95342 1/20 0.45
NR3C1 P04150 1/20 0.45
CHRM2 P08172 1/20 0.45
HTR1A P08908 1/20 0.45
ADRA2A P08913 1/20 0.45
ADORA3 P0DMS8 1/20 0.45
CHRM1 P11229 1/20 0.45
DRD2 P14416 1/20 0.45
ADRA2B P18089 1/20 0.45
ADRA2C P18825 1/20 0.45
DRD1 P21728 1/20 0.45
SLC6A2 P23975 1/20 0.45
HTR2A P28223 1/20 0.45
SLC6A4 P31645 1/20 0.45
ADRA1A P35348 1/20 0.45
PTGS2 P35354 1/20 0.45
OPRM1 P35372 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7576311 0.99 ESR1 (0.61) ESR1ESR2MLNRABCB11NR3C1
SCHEMBL8504438 0.95 ESR1 (0.55) ESR1ESR2MLNRABCB11NR3C1
SCHEMBL7574747 0.90 ESR1 (0.73) ESR1ESR2
SCHEMBL7576301 0.89 ESR1 (0.74) ESR1ESR2
SCHEMBL7571727 0.89 LTA4H (0.51) ESR1ESR2HRH3
SCHEMBL7582532 0.88 ESR1 (0.65) ESR1ESR2
SCHEMBL7574347 0.88 LTA4H (0.52) ESR1ESR2HRH3
SCHEMBL7580135 0.88 ESR1 (0.67) ESR1ESR2
SCHEMBL7574693 0.87 ESR1 (0.61) ESR1ESR2
SCHEMBL7580940 0.86 ESR1 (0.64) ESR1ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5994370-A ESTROGEN RECEPTOR MODULATORS ELI LILLY AND COMPANY (US) 1999-11-30 US claimed
EP-0873992-B1 Indene compounds having activity as SERMs LILLY CO ELI (US) 2002-09-25 EP disclosed
US-5994370-A ESTROGEN RECEPTOR MODULATORS ELI LILLY AND COMPANY (US) 1999-11-30 US disclosed
EP-0873992-A1 Indene compounds having activity as SERMs ELI LILLY AND COMPANY (US) 1998-10-28 EP disclosed