SCHEMBL7573148

SCHEMBL7573148

O=[N+]([O-])c1ccc(C#CCN=Cc2ccc([N+](=O)[O-])cc2)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIN2D O15399 2/20 0.44
GRIN3B O60391 2/20 0.44
GRIN1 Q05586 2/20 0.44
GRIN2A Q12879 2/20 0.44
GRIN2B Q13224 2/20 0.44
GRIN2C Q14957 2/20 0.44
GRIN3A Q8TCU5 2/20 0.44
CTDSP1 Q9GZU7 1/20 0.43
AMY1A P0DUB6 1/20 0.43
NPC1 O15118 4/20 0.42
MAPT P10636 5/20 0.41
MAOB P27338 1/20 0.41
APP P05067 1/20 0.41
PTGS2 P35354 2/20 0.40
CA12 O43570 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CA9 Q16790 1/20 0.40
FBP1 P09467 1/20 0.40
CASP3 P42574 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7573146 1.00 GRIN2D (0.44) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL7571219 0.93 ACHE (0.47) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL7572697 0.93 MAPT (0.45) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL7572694 0.93 MAPT (0.45) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL7581527 0.93 MEN1 (0.49) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL7579070 0.93 MEN1 (0.49) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL7579065 0.93 MEN1 (0.49) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL7581536 0.93 MEN1 (0.49) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL7580865 0.90 MEN1 (0.49) MAPTMAOBAPPPTGS2ALDH1A1
SCHEMBL7572281 0.86 MEN1 (0.51) AMY1ANPC1MAPTPTGS2CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0810199-B1 Method for producing propargylamine compounds SUMITOMO CHEMICAL CO (JP) 2002-09-25 EP disclosed
US-5756769-A Method for producing propargylamine compounds SUMITOMO CHEMICAL COMPANY, LTD. (JP) 1998-05-26 US disclosed
EP-0810199-A1 Method for producing propargylamine compounds SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1997-12-03 EP disclosed