SCHEMBL7573409

SCHEMBL7573409

Cc1ccc(C#CC/N=C/c2cccc(Cl)c2)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM5 P08912 1/20 0.45
MAPT P10636 5/20 0.40
GAA P10253 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.39
GRIN2D O15399 2/20 0.38
GRIN3B O60391 2/20 0.38
GRIN1 Q05586 2/20 0.38
GRIN2A Q12879 2/20 0.38
GRIN2B Q13224 2/20 0.38
GRIN2C Q14957 2/20 0.38
GRIN3A Q8TCU5 2/20 0.38
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
CYP1A2 P05177 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C19 P33261 1/20 0.38
ALOX5 P09917 1/20 0.36
NPC1 O15118 3/20 0.36
ALDH1A1 P00352 3/20 0.36
RAB9A P51151 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7573410 1.00 CHRM5 (0.45) CHRM5MAPTGAASMN1; SMN2GRIN2D
SCHEMBL7578981 0.87 CHRM5 (0.49) CHRM5MAPTGAASMN1; SMN2GRIN2D
SCHEMBL7578987 0.87 CHRM5 (0.49) CHRM5MAPTGAASMN1; SMN2GRIN2D
SCHEMBL7571676 0.86 CHRM5 (0.50) CHRM5MAPTGAASMN1; SMN2GRIN2D
SCHEMBL7571671 0.86 CHRM5 (0.50) CHRM5MAPTGAASMN1; SMN2GRIN2D
SCHEMBL7573181 0.86 RELA (0.51) CHRM5MAPTGAAALOX5NPC1
SCHEMBL7573177 0.86 RELA (0.51) CHRM5MAPTGAAALOX5NPC1
SCHEMBL7572816 0.83 CHRM5 (0.42) CHRM5MAPTGAASMN1; SMN2GRIN2D
SCHEMBL7572820 0.83 CHRM5 (0.42) CHRM5MAPTGAASMN1; SMN2GRIN2D
SCHEMBL7579764 0.83 NPC1 (0.39) MAPTSMN1; SMN2MEN1KMT2ACYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0810199-B1 Method for producing propargylamine compounds SUMITOMO CHEMICAL CO (JP) 2002-09-25 EP disclosed
US-5756769-A Method for producing propargylamine compounds SUMITOMO CHEMICAL COMPANY, LTD. (JP) 1998-05-26 US disclosed
EP-0810199-A1 Method for producing propargylamine compounds SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1997-12-03 EP disclosed