SCHEMBL7573181

SCHEMBL7573181

COc1ccc(C#CCN=Cc2cccc(Cl)c2)cc1

nearest known ligand 0.51

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
RELA Q04206 1/20 0.51
MAPT P10636 2/20 0.43
NFE2L2 Q16236 2/20 0.43
TP53 P04637 1/20 0.43
CHRM5 P08912 2/20 0.42
AHR P35869 1/20 0.38
XDH P47989 2/20 0.38
GAA P10253 1/20 0.38
EGFR P00533 1/20 0.37
KCNH2 Q12809 1/20 0.37
GSK3B P49841 1/20 0.37
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
ALOX5 P09917 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7573177 1.00 RELA (0.51) RELAMAPTNFE2L2TP53CHRM5
SCHEMBL7573409 0.86 CHRM5 (0.45) MAPTCHRM5GAAKCNH2NPC1
SCHEMBL7573410 0.86 CHRM5 (0.45) MAPTCHRM5GAAKCNH2NPC1
SCHEMBL7572532 0.84 MAOB (0.39) RELAMAPTNFE2L2TP53AHR
SCHEMBL7572529 0.84 MAOB (0.39) RELAMAPTNFE2L2TP53AHR
SCHEMBL7579606 0.84 TRPA1 (0.45) MAPTGAAKCNH2NPC1RAB9A
SCHEMBL7578987 0.84 CHRM5 (0.49) MAPTCHRM5GAANPC1RAB9A
SCHEMBL7578981 0.84 CHRM5 (0.49) MAPTCHRM5GAANPC1RAB9A
SCHEMBL7579599 0.84 TRPA1 (0.45) MAPTGAAKCNH2NPC1RAB9A
SCHEMBL7571671 0.83 CHRM5 (0.50) MAPTCHRM5GAAKCNH2NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0810199-B1 Method for producing propargylamine compounds SUMITOMO CHEMICAL CO (JP) 2002-09-25 EP disclosed
US-5756769-A Method for producing propargylamine compounds SUMITOMO CHEMICAL COMPANY, LTD. (JP) 1998-05-26 US disclosed
EP-0810199-A1 Method for producing propargylamine compounds SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1997-12-03 EP disclosed