SCHEMBL7572816

SCHEMBL7572816

Cc1ccc(C#CC/N=C/c2cccc(Cl)c2)c(C)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM5 P08912 1/20 0.42
SMN1; SMN2 Q16637 3/20 0.37
GRIN2D O15399 2/20 0.36
GRIN3B O60391 2/20 0.36
GRIN1 Q05586 2/20 0.36
GRIN2A Q12879 2/20 0.36
GRIN2B Q13224 2/20 0.36
GRIN2C Q14957 2/20 0.36
GRIN3A Q8TCU5 2/20 0.36
NPC1 O15118 5/20 0.36
CASP3 P42574 1/20 0.36
SENP8 Q96LD8 1/20 0.36
SENP7 Q9BQF6 1/20 0.36
SENP6 Q9GZR1 1/20 0.36
MAPT P10636 4/20 0.35
KMT2A Q03164 2/20 0.35
MEN1 O00255 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C19 P33261 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7572820 1.00 CHRM5 (0.42) CHRM5SMN1; SMN2GRIN2DGRIN3BGRIN1
SCHEMBL7574195 0.87 CHRM5 (0.44) CHRM5SMN1; SMN2GRIN2DGRIN3BGRIN1
SCHEMBL7574192 0.87 CHRM5 (0.44) CHRM5SMN1; SMN2GRIN2DGRIN3BGRIN1
SCHEMBL7580233 0.86 PARP15 (0.38) SMN1; SMN2NPC1KMT2AMEN1CYP1A2
SCHEMBL7580227 0.86 PARP15 (0.38) SMN1; SMN2NPC1KMT2AMEN1CYP1A2
SCHEMBL7575405 0.85 NFE2L2 (0.35) SMN1; SMN2NPC1CASP3SENP8SENP7
SCHEMBL7575413 0.85 NFE2L2 (0.35) SMN1; SMN2NPC1CASP3SENP8SENP7
SCHEMBL7573409 0.83 CHRM5 (0.45) CHRM5SMN1; SMN2GRIN2DGRIN3BGRIN1
SCHEMBL7573410 0.83 CHRM5 (0.45) CHRM5SMN1; SMN2GRIN2DGRIN3BGRIN1
SCHEMBL7571852 0.80 NFE2L2 (0.47) SMN1; SMN2KMT2AMEN1CYP1A2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0810199-B1 Method for producing propargylamine compounds SUMITOMO CHEMICAL CO (JP) 2002-09-25 EP disclosed
US-5756769-A Method for producing propargylamine compounds SUMITOMO CHEMICAL COMPANY, LTD. (JP) 1998-05-26 US disclosed
EP-0810199-A1 Method for producing propargylamine compounds SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1997-12-03 EP disclosed