SCHEMBL7573483

SCHEMBL7573483

Clc1ccc(C=NCC#Cc2ccc(Br)s2)cc1

nearest known ligand 0.34

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MAOB P27338 1/20 0.34
CYP1A2 P05177 1/20 0.33
TSHR P16473 1/20 0.33
ADORA2A P29274 1/20 0.30
ADORA1 P30542 1/20 0.30
GRIN2D O15399 1/20 0.30
GRIN3B O60391 1/20 0.30
GRIN1 Q05586 1/20 0.30
GRIN2A Q12879 1/20 0.30
GRIN2B Q13224 1/20 0.30
GRIN2C Q14957 1/20 0.30
GRIN3A Q8TCU5 1/20 0.30
G6PC1 P35575 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7573127 0.86 CA2 (0.33)
SCHEMBL7573124 0.86 CA2 (0.33)
SCHEMBL7579771 0.81 MAPT (0.40) MAOBGRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL7573394 0.78 GRIN2D (0.33) CYP1A2GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL7575258 0.74 G6PC1 (0.35) ADORA1G6PC1
SCHEMBL7575256 0.74 G6PC1 (0.35) ADORA1G6PC1
SCHEMBL7571802 0.73 G6PC1 (0.36) MAOBCYP1A2TSHRGRIN2DGRIN3B
SCHEMBL7579060 0.72 G6PC1 (0.43) MAOBCYP1A2GRIN1GRIN2BG6PC1
SCHEMBL7579055 0.72 G6PC1 (0.43) MAOBCYP1A2GRIN1GRIN2BG6PC1
SCHEMBL7575202 0.71 MAOB (0.44) MAOBCYP1A2TSHRADORA2AADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0810199-B1 Method for producing propargylamine compounds SUMITOMO CHEMICAL CO (JP) 2002-09-25 EP disclosed
US-5756769-A Method for producing propargylamine compounds SUMITOMO CHEMICAL COMPANY, LTD. (JP) 1998-05-26 US disclosed
EP-0810199-A1 Method for producing propargylamine compounds SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1997-12-03 EP disclosed