SCHEMBL7573850

SCHEMBL7573850

Nc1cc(N2CCCCC2)ncc1C(=O)N1CCCCC1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.46
HPGD P15428 4/20 0.46
KDM4E B2RXH2 3/20 0.46
POLB P06746 2/20 0.46
ALOX15 P16050 1/20 0.46
HSD17B10 Q99714 1/20 0.46
HSD11B1 P28845 1/20 0.41
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
ADORA2A P29274 1/20 0.40
HSP90AA1 P07900 1/20 0.40
LMNA P02545 2/20 0.40
TP53 P04637 2/20 0.40
GBA1 P04062 2/20 0.39
L3MBTL3 Q96JM7 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
CYP2C9 P11712 1/20 0.39
TSHR P16473 1/20 0.39
PIK3C3 Q8NEB9 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20089110 0.76 CNR2 (0.46) ALDH1A1KMT2ALMNANPSR1TSHR
SCHEMBL25855482 0.74 CNR2 (0.43) ALDH1A1KDM4EKMT2ALMNANPSR1
SCHEMBL26088188 0.74 KDM4E (0.46) ALDH1A1KDM4EPOLBALOX15HSD17B10
SCHEMBL30280743 0.73 CNR2 (0.44) ALDH1A1KMT2ALMNANPSR1TSHR
SCHEMBL12488177 0.73 CNR2 (0.44) ALDH1A1KMT2ALMNANPSR1TSHR
SCHEMBL21262379 0.71 AR (0.44) ALDH1A1KMT2ALMNANPSR1TSHR
SCHEMBL17774955 0.71 HSD11B1 (0.51) ALDH1A1HPGDKDM4EPOLBHSD17B10
SCHEMBL17774959 0.71 ALDH1A1 (0.46) ALDH1A1HPGDKDM4EPOLBHSD17B10
SCHEMBL25958653 0.70 ALDH1A1 (0.42) ALDH1A1HPGDKDM4EHSD11B1MEN1
SCHEMBL3899784 0.70 L3MBTL3 (0.54) ALDH1A1HPGDKDM4EPOLBALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1242404-A1 PHENOXYPROPANOLAMINES, PREPARATION AND THERAPEUTIC USE THEREOF SANOFI-SYNTHELABO (FR) 2002-09-25 EP disclosed
WO-2001044227-A1 PHENOXYPROPANOLAMINES, PREPARATION AND THERAPEUTIC USE THEREOF SANOFI-SYNTHELABO (FR) 2001-06-21 WO disclosed