SCHEMBL7573969

SCHEMBL7573969

Cc1ccc(Cl)c2cc3cccc(C(=O)O)c3nc12

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PPARA Q07869 1/20 0.43
KDM4E B2RXH2 2/20 0.42
LMNA P02545 2/20 0.42
HTT P42858 1/20 0.42
ACLY P53396 1/20 0.41
MEN1 O00255 4/20 0.41
KMT2A Q03164 4/20 0.41
ALDH1A1 P00352 2/20 0.41
GLA P06280 1/20 0.41
PKM P14618 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
NPY1R P25929 1/20 0.41
NPY2R P49146 1/20 0.41
NR4A1 P22736 2/20 0.40
NR4A2 P43354 2/20 0.40
AKR1B10 O60218 1/20 0.40
ABCB11 O95342 1/20 0.40
TTR P02766 1/20 0.40
ADORA3 P0DMS8 1/20 0.40
CHRM1 P11229 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7567029 0.89 RAD52 (0.45) PPARAKDM4ELMNAHTTMEN1
SCHEMBL7568079 0.88 ALDH1A1 (0.51) KDM4ELMNAHTTACLYMEN1
SCHEMBL5459806 0.81 ALDH1A1 (0.50) KDM4ELMNAHTTKMT2AALDH1A1
SCHEMBL7564788 0.78 KDM4E (0.47) KDM4ELMNAHTTMEN1KMT2A
SCHEMBL7623210 0.78 ALDH1A1 (0.44) KDM4ELMNAHTTACLYMEN1
SCHEMBL1906559 0.78 TSHR (0.44) PPARAKDM4ELMNAACLYMEN1
SCHEMBL7567221 0.77 TSHR (0.52) KDM4ELMNAMEN1KMT2AALDH1A1
SCHEMBL7565057 0.76 RAD52 (0.54) HTT
SCHEMBL7569010 0.76 ALDH1A1 (0.58) PPARAKDM4ELMNAACLYMEN1
SCHEMBL7565052 0.75 RAD52 (0.46) KDM4EMEN1KMT2AALDH1A1GLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1116285-C Bis(acridinecarboxamide) and Bis(phenazinecarboxamide) as antitumour agents XENOVA LTD (GB) 2003-07-30 CN disclosed
EP-0934278-B1 BIS(ACRIDINECARBOXAMIDE) AND BIS(PHENAZINECARBOXAMIDE) AS ANTITUMOUR AGENTS XENOVA LTD (GB) 2002-09-04 EP disclosed
US-6114332-A BACTERICIDES XENOVA LIMITED (GB) 2000-09-05 US disclosed
CN-1240430-A Bis(acridinecarboxamide) and Bis(phenazinecarboxamide) as antitumour agents XENOVA LTD (GB) 2000-01-05 CN disclosed
EP-0934278-A1 BIS(ACRIDINECARBOXAMIDE) AND BIS(PHENAZINECARBOXAMIDE) AS ANTITUMOUR AGENTS XENOVA LIMITED (GB) 1999-08-11 EP disclosed
WO-1998017650-A1 BIS(ACRIDINECARBOXAMIDE) AND BIS(PHENAZINECARBOXAMIDE) AS ANTITUMOUR AGENTS XENOVA LIMITED (GB) 1998-04-30 WO disclosed