SCHEMBL7575808

SCHEMBL7575808

O=C1N=C(O)C(c2ccc(C(F)(F)F)cc2)=NC1Cc1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CES2 O00748 1/20 0.41
CCKAR P32238 3/20 0.38
CCKBR P32239 3/20 0.38
KIF11 P52732 1/20 0.37
BACE1 P56817 1/20 0.37
CFTR P13569 1/20 0.37
LMNA P02545 1/20 0.35
HTT P42858 1/20 0.35
BDKRB2 P30411 1/20 0.35
HDAC3 O15379 1/20 0.35
HDAC1 Q13547 1/20 0.35
HDAC8 Q9BY41 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
PTPN2 P17706 1/20 0.34
PTPN1 P18031 1/20 0.34
PTPN6 P29350 1/20 0.34
TP53 P04637 1/20 0.34
GLO1 Q04760 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7570328 0.95 CES2 (0.45) CES2CCKARCCKBRKIF11BACE1
SCHEMBL7572646 0.87 BDKRB2 (0.41) CES2LMNAHTTBDKRB2HDAC3
SCHEMBL7572458 0.87 BDKRB2 (0.42) CES2BDKRB2HDAC3HDAC1HDAC8
SCHEMBL7571711 0.86 CES2 (0.38) CES2CCKARCCKBRLMNABDKRB2
SCHEMBL7571381 0.86 HDAC3 (0.42) CCKARCCKBRBDKRB2HDAC3HDAC1
SCHEMBL7571208 0.84 NPC1 (0.44) CES2BDKRB2HDAC3HDAC1HDAC8
SCHEMBL7576544 0.84 CES2 (0.44) CES2LMNABDKRB2HDAC3HDAC1
SCHEMBL7572631 0.81 CES2 (0.42) CES2CCKARCCKBRBDKRB2HDAC3
SCHEMBL7572718 0.79 CES2 (0.43) CES2LMNABDKRB2HDAC3HDAC1
SCHEMBL7570886 0.78 PSD (0.37) HTTBDKRB2HDAC3HDAC1HDAC8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002085369-A1 INHIBITORS OF ANTHRAX LETHAL FACTOR ACTIVITY STRUCTURAL BIOINFORMATICS, INC. (US) 2002-10-31 WO disclosed