SCHEMBL7578013

SCHEMBL7578013

O=C1N=C(O)C(c2ccc(N3CCOCC3)cc2)=NC1Cc1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 3/20 0.43
MAPT P10636 4/20 0.41
LMNA P02545 2/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
TSHR P16473 2/20 0.40
PKM P14618 1/20 0.40
PIK3C3 Q8NEB9 5/20 0.39
ATM Q13315 5/20 0.39
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
POLB P06746 1/20 0.39
HSP90AA1 P07900 1/20 0.39
HSP90AB1 P08238 1/20 0.39
GAA P10253 1/20 0.39
ALOX15 P16050 1/20 0.39
ALOX12 P18054 1/20 0.39
MAPK1 P28482 1/20 0.39
RECQL P46063 1/20 0.39
TDP1 Q9NUW8 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7577759 0.96 MAPT (0.40) KIF11MAPTLMNASMN1; SMN2L3MBTL1
SCHEMBL7572646 0.82 BDKRB2 (0.41) LMNATSHRGAA
SCHEMBL7572458 0.82 BDKRB2 (0.42)
SCHEMBL7571381 0.81 HDAC3 (0.42)
SCHEMBL7576544 0.79 CES2 (0.44) MAPTLMNAKDM4EALDH1A1
SCHEMBL7571711 0.79 CES2 (0.38) LMNA
SCHEMBL7571208 0.79 NPC1 (0.44) MAPTSMN1; SMN2ALDH1A1POLBGAA
SCHEMBL7569645 0.76 DHODH (0.38) MAPTHSP90AA1GAATDP1
SCHEMBL7572631 0.75 CES2 (0.42) SMN1; SMN2ALDH1A1GAA
SCHEMBL7572718 0.75 CES2 (0.43) MAPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002085369-A1 INHIBITORS OF ANTHRAX LETHAL FACTOR ACTIVITY STRUCTURAL BIOINFORMATICS, INC. (US) 2002-10-31 WO disclosed