SCHEMBL7579146

SCHEMBL7579146

C#C/C(N)=C\c1cccc(OC)c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 1/20 0.51
MEN1 O00255 1/20 0.49
ALDH1A1 P00352 1/20 0.49
KMT2A Q03164 1/20 0.49
CHRM5 P08912 1/20 0.49
CYP19A1 P11511 1/20 0.47
NQO2 P16083 1/20 0.47
RELA Q04206 1/20 0.47
MAPT P10636 2/20 0.46
FOS P01100 1/20 0.46
JUN P05412 1/20 0.46
NFE2L2 Q16236 2/20 0.45
KDM4E B2RXH2 1/20 0.44
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
PARP1 P09874 1/20 0.44
PRSS1 P07477 1/20 0.44
PRSS2 P07478 1/20 0.44
PRSS3 P35030 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15286598 0.84 MAPT (0.53) TAAR1MEN1ALDH1A1KMT2ACHRM5
SCHEMBL7581521 0.80 ALDH1A1 (0.53) ALDH1A1NQO2MAPTKDM4ERAB9A
SCHEMBL22791460 0.80 TAAR1 (0.57) TAAR1MEN1ALDH1A1KMT2ACHRM5
SCHEMBL7572617 0.78 TP53 (0.46) MEN1ALDH1A1KMT2ARELAMAPT
SCHEMBL14198012 0.75 CHRM5 (0.58) TAAR1MEN1ALDH1A1KMT2ACHRM5
SCHEMBL9416087 0.75 TAAR1 (0.53) TAAR1MEN1ALDH1A1KMT2ACHRM5
SCHEMBL19901437 0.75 MEN1 (0.54) TAAR1MEN1ALDH1A1KMT2ACHRM5
SCHEMBL7572362 0.75 MAOB (0.49) CHRM5NQO2MAPTNFE2L2NPC1
SCHEMBL7575017 0.75 GRIN1 (0.47) MEN1ALDH1A1KMT2ACHRM5MAPT
SCHEMBL10689025 0.74 MEN1 (0.64) TAAR1MEN1ALDH1A1KMT2ACHRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0810199-B1 Method for producing propargylamine compounds SUMITOMO CHEMICAL CO (JP) 2002-09-25 EP disclosed
US-5756769-A Method for producing propargylamine compounds SUMITOMO CHEMICAL COMPANY, LTD. (JP) 1998-05-26 US disclosed
EP-0810199-A1 Method for producing propargylamine compounds SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1997-12-03 EP disclosed