SCHEMBL7575017

SCHEMBL7575017

C#C/C(N)=C\c1cccc(Cl)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIN1 Q05586 4/20 0.47
GRIN2B Q13224 4/20 0.47
GRIN2D O15399 2/20 0.47
GRIN3B O60391 2/20 0.47
GRIN2A Q12879 2/20 0.47
GRIN2C Q14957 2/20 0.47
GRIN3A Q8TCU5 2/20 0.47
CYP1A2 P05177 2/20 0.47
CYP2C9 P11712 1/20 0.47
FBP1 P09467 2/20 0.46
GAA P10253 1/20 0.45
MAPT P10636 1/20 0.45
CHRM5 P08912 1/20 0.44
KMT2A Q03164 2/20 0.43
KDM4E B2RXH2 1/20 0.43
ALDH1A1 P00352 1/20 0.43
POLB P06746 1/20 0.43
PKM P14618 1/20 0.43
KIF20A O95235 1/20 0.40
PARP1 P09874 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28459287 0.82 MAPT (0.56) GRIN1GRIN2BGRIN2DGRIN3BGRIN2A
SCHEMBL7573585 0.79 HSD17B3 (0.47) MAPTKMT2AALDH1A1POLBPKM
SCHEMBL7572362 0.79 MAOB (0.49) CYP1A2FBP1MAPTCHRM5PKM
SCHEMBL7572617 0.79 TP53 (0.46) CYP1A2FBP1GAAMAPTKMT2A
SCHEMBL7575165 0.77 GRIN2D (0.41) GRIN1GRIN2BGRIN2DGRIN3BGRIN2A
SCHEMBL7572848 0.77 MCL1 (0.46) GRIN1GRIN2BGRIN2DGRIN3BGRIN2A
SCHEMBL7579146 0.75 TAAR1 (0.51) MAPTCHRM5KMT2AKDM4EALDH1A1
SCHEMBL7573955 0.72 FBP1 (0.57) CYP1A2FBP1MAPTKMT2AKDM4E
SCHEMBL6867023 0.71 GRIN2B (0.47) GRIN1GRIN2BGRIN2DGRIN3BGRIN2A
SCHEMBL7573441 0.71 GABRA1 (0.51) GRIN1GRIN2BGRIN2DGRIN3BGRIN2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0810199-B1 Method for producing propargylamine compounds SUMITOMO CHEMICAL CO (JP) 2002-09-25 EP disclosed
US-5756769-A Method for producing propargylamine compounds SUMITOMO CHEMICAL COMPANY, LTD. (JP) 1998-05-26 US disclosed
EP-0810199-A1 Method for producing propargylamine compounds SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1997-12-03 EP disclosed