SCHEMBL7582780

SCHEMBL7582780

C=CCc1cc(Br)cc(Br)c1O

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.50
TSHR P16473 1/20 0.50
TDP1 Q9NUW8 1/20 0.50
GABRA1 P14867 3/20 0.45
GABRB2 P47870 3/20 0.45
GABRB1 P18505 1/20 0.45
GABRA2 P47869 1/20 0.45
GFER P55789 1/20 0.44
KMT2A Q03164 6/20 0.42
MEN1 O00255 5/20 0.42
MAPT P10636 5/20 0.42
ALDH1A1 P00352 1/20 0.42
POLB P06746 1/20 0.42
PLEC Q15149 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C19 P33261 1/20 0.42
HIF1A Q16665 1/20 0.42
ERN1 O75460 1/20 0.42
LMNA P02545 3/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL930281 0.81 ERN1 (0.46) GABRA1GABRB2KMT2AMEN1MAPT
SCHEMBL14742304 0.81 GABRA1 (0.39) GABRA1GABRB2GFERKMT2AMEN1
SCHEMBL4233697 0.81 GABRA1 (0.39) CYP3A4GABRA1GABRB2KMT2AMEN1
SCHEMBL4219327 0.81 GAA (0.43) GABRA1GABRB2KMT2AMEN1MAPT
SCHEMBL4230006 0.81 GABRA1 (0.39) CYP3A4TSHRTDP1GABRA1GABRB2
SCHEMBL333372 0.81 ALOX5 (0.47) GABRA1GABRB2KMT2AMEN1MAPT
SCHEMBL1620174 0.80 GAA (0.51) CYP3A4TSHRGABRA1GABRB2KMT2A
SCHEMBL3658549 0.80 ERN1 (0.52) CYP3A4TSHRTDP1GABRA1GABRB2
SCHEMBL1003056 0.78 KDM4E (0.61) CYP3A4TDP1GABRA1GABRB2KMT2A
SCHEMBL1360502 0.78 ERN1 (0.55) GABRA1GABRB2KMT2AMEN1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1228055-A1 DIHYDROAMINOBENZO[B]- AND [C]FURANS AS RETINOID-LIKE AGENTS Allergan Sales, Inc. (US) 2002-08-07 EP disclosed
WO-2001012618-A1 DIHYDROAMINOBENZO[B]- AND [C]FURANS AS RETINOID-LIKE AGENTS ALLERGAN SALES, INC. (US) 2001-02-22 WO disclosed
US-6093838-A FOR TREATING SKIN-RELATED DISEASES, INCLUDING ACTINIC KERATOSES, ARSENIC KERATOSES, ECZEMA ALLERGAN SALES, INC. (US) 2000-07-25 US disclosed