SCHEMBL7583086

SCHEMBL7583086

COc1ccc(C(C)(C)CC#N)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.43
GAA P10253 2/20 0.43
CA12 O43570 1/20 0.42
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
CA7 P43166 1/20 0.42
CA9 Q16790 1/20 0.42
CA14 Q9ULX7 1/20 0.42
HSD17B10 Q99714 2/20 0.41
APEX1 P27695 2/20 0.41
LMNA P02545 1/20 0.41
ALOX15 P16050 1/20 0.41
MAPK1 P28482 1/20 0.41
RECQL P46063 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
AOC3 Q16853 1/20 0.41
PBRM1 Q86U86 1/20 0.39
MAPT P10636 3/20 0.39
CASP1 P29466 1/20 0.38
KDM4E B2RXH2 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8558744 0.79 LMNA (0.44) ALDH1A1GAACA12CA1CA2
SCHEMBL9447336 0.78 TSHR (0.46) ALDH1A1GAACA1CA2CA9
SCHEMBL20782023 0.78 APP (0.47) ALDH1A1GAAHSD17B10APEX1LMNA
Acetonitrile SCHEMBL8561616 0.77 LMNA (0.42) ALDH1A1GAACA12CA1CA2
SCHEMBL6801469 0.77 AOC3 (0.41) ALDH1A1GAACA12CA1CA2
SCHEMBL2815949 0.76 MAPT (0.47) ALDH1A1MAPK1MAPTCYP1A2CYP3A4
SCHEMBL3045851 0.76 CYP2A6 (0.33) ALDH1A1CA1CA2CA9HSD17B10
SCHEMBL3436081 0.75 NPC1 (0.60) ALDH1A1CA12CA1CA2CA7
SCHEMBL1506598 0.75 CA1 (0.50) ALDH1A1CA12CA1CA2CA7
SCHEMBL4673742 0.75 TAAR1 (0.52) ALDH1A1ALOX15MAPK1MAPTCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0780375-B1 3-((5-substituted benzyl)amino)-2-phenylpiperidines as substance p antagonists PFIZER (US) 2002-09-11 EP disclosed
US-5789423-A ANTIALLERGENS, ANTIINFLAMMATORY AGENTS; GASTROINTESTINAL AND CENTRAL NERVOUS SYSTEM DISORDERS PFIZER INC. (US) 1998-08-04 US disclosed
EP-0780375-A1 3-((5-substituted benzyl)amino)-2-phenylpiperidines as substance p antagonists PFIZER INC. (US) 1997-06-25 EP disclosed