SCHEMBL7585541

SCHEMBL7585541

CC(C)CCC(=O)N[C@@H](CC1CCCCC1)C(=O)N(C)C#N

nearest known ligand 0.50

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CTSK P43235 13/20 0.50
CTSL P07711 8/20 0.46
CTSB P07858 8/20 0.46
CTSH P09668 5/20 0.46
CTSS P25774 3/20 0.43
CTSD P07339 1/20 0.40
PSEN1 P49768 4/20 0.39
PSEN2 P49810 4/20 0.39
APH1B Q8WW43 4/20 0.39
NCSTN Q92542 4/20 0.39
APH1A Q96BI3 4/20 0.39
PSENEN Q9NZ42 4/20 0.39
CHRNB2 P17787 1/20 0.38
CHRNB4 P30926 1/20 0.38
CHRNA3 P32297 1/20 0.38
CHRNA4 P43681 1/20 0.38
GRIN1 Q05586 1/20 0.38
GRIN2A Q12879 1/20 0.38
GRM1 Q13255 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5528178 0.87 CTSK (0.48) CTSKCTSLCTSBCTSHCTSS
SCHEMBL5527109 0.87 CTSK (0.48) CTSKCTSLCTSBCTSHCTSS
SCHEMBL5523001 0.83 CTSK (0.51) CTSKCTSLCTSBCTSHCTSS
SCHEMBL5526860 0.82 CTSK (0.50) CTSKCTSLCTSBCTSHCTSS
SCHEMBL5529190 0.80 CTSL (0.48) CTSKCTSLCTSBCTSHCTSS
SCHEMBL5528340 0.80 CTSL (0.48) CTSKCTSLCTSBCTSHCTSS
SCHEMBL5527441 0.80 CTSK (0.61) CTSKCTSLCTSBCTSHCTSS
SCHEMBL5523059 0.77 CTSS (0.53) CTSKCTSLCTSBCTSHCTSS
SCHEMBL5525335 0.74 CTSL (0.69) CTSKCTSLCTSBCTSSCHRNB2
SCHEMBL5530441 0.74 CTSL (0.69) CTSKCTSLCTSBCTSSCHRNB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1178958-A2 N-CYANOMETHYL AMIDES AS PROTEASE INHIBITORS AXYS PHARMACEUTICALS, INC. (US) 2002-02-13 EP disclosed
WO-2000055125-A2 N-CYANOMETHYL AMIDES AS PROTEASE INHIBITORS AXYS PHARMACEUTICALS, INC. (US) 2000-09-21 WO disclosed