SCHEMBL7586310

SCHEMBL7586310

CCN1CCC2(CCc3ccccc3C2=O)CC1.O=C1c2ccccc2CCC12CCN(C/C=C/c1ccccc1)CC2

nearest known ligand 0.58

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 15/20 0.58
HTR2A P28223 12/20 0.58
HTR2C P28335 12/20 0.58
HTR2B P41595 12/20 0.58
DRD2 P14416 12/20 0.58
ALDH1A1 P00352 1/20 0.46
MAPT P10636 1/20 0.46
KDM4E B2RXH2 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6836323 0.94 SIGMAR1 (0.64) SIGMAR1HTR2AHTR2CHTR2BDRD2
SCHEMBL6836322 0.94 SIGMAR1 (0.64) SIGMAR1HTR2AHTR2CHTR2BDRD2
SCHEMBL7587346 0.86 SIGMAR1 (0.73) SIGMAR1HTR2AHTR2CHTR2BDRD2
SCHEMBL6843243 0.82 SIGMAR1 (0.55) SIGMAR1HTR2AHTR2CHTR2BDRD2
SCHEMBL6841101 0.82 DRD2 (0.55) SIGMAR1HTR2AHTR2CHTR2BDRD2
SCHEMBL6840814 0.82 SIGMAR1 (0.66) SIGMAR1HTR2AHTR2CHTR2BDRD2
SCHEMBL6836327 0.78 KDM4E (0.45) SIGMAR1HTR2AHTR2CHTR2BDRD2
SCHEMBL6840845 0.78 SIGMAR1 (0.66) SIGMAR1HTR2AHTR2CHTR2BDRD2
SCHEMBL14045655 0.75 ALDH1A1 (0.63) SIGMAR1HTR2AHTR2CHTR2BDRD2
SCHEMBL6841555 0.75 ALDH1A1 (0.47) SIGMAR1HTR2AHTR2BDRD2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1235808-A2 TRICYCLIC ANALGESICS WARNER-LAMBERT COMPANY (US) 2002-09-04 EP claimed
WO-2000075116-A2 TRICYCLIC ANALGESICS WARNER-LAMBERT COMPANY (US) 2000-12-14 WO claimed