SCHEMBL7588071

SCHEMBL7588071

CN(C)CC1=C(c2cccc(O)c2)c2ccc(-c3cccc(O)c3)cc2CC1

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TDP2 O95551 1/20 0.41
HSD17B1 P14061 10/20 0.41
HSD17B2 P37059 8/20 0.41
CYP3A4 P08684 2/20 0.41
CYP2C9 P11712 2/20 0.41
OPRK1 P41145 1/20 0.41
ESR1 P03372 4/20 0.38
ADORA1 P30542 1/20 0.37
OPRD1 P41143 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2B6 P20813 1/20 0.36
CYP2C19 P33261 1/20 0.36
ESR2 Q92731 1/20 0.36
PRF1 P14222 1/20 0.36
PIM1 P11309 1/20 0.36
PIM2 Q9P1W9 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8012237 0.99 TDP2 (0.40) TDP2HSD17B1HSD17B2CYP3A4CYP2C9
SCHEMBL7587708 0.96 OPRK1 (0.46) TDP2HSD17B1HSD17B2CYP3A4CYP2C9
Hydrochloric Acid SCHEMBL8013584 0.95 OPRK1 (0.45) TDP2HSD17B1HSD17B2CYP3A4CYP2C9
SCHEMBL7588665 0.93 ESR1 (0.40) HSD17B1HSD17B2ESR1ESR2
SCHEMBL7586120 0.93 TAAR1 (0.41) TDP2HSD17B1HSD17B2CYP3A4CYP2C9
SCHEMBL7586132 0.93 TAAR1 (0.47) TDP2HSD17B1HSD17B2CYP3A4CYP2C9
Hydrochloric Acid SCHEMBL8017994 0.92 ESR1 (0.39) HSD17B1HSD17B2ESR1ESR2
Hydrochloric Acid SCHEMBL8014418 0.92 TAAR1 (0.46) TDP2HSD17B1HSD17B2CYP3A4CYP2C9
Hydrochloric Acid SCHEMBL8011965 0.92 AOC3 (0.41) TDP2HSD17B1HSD17B2CYP3A4CYP2C9
SCHEMBL7591741 0.88 MTNR1A (0.44) TDP2HSD17B1HSD17B2CYP3A4OPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0864559-B1 Substituted amino compounds and their use as analgesic active substances GRUENENTHAL GMBH (DE) 2002-06-05 EP disclosed
EP-0864559-A1 Substituted amino compounds and their use as analgesic active substances Grünenthal GmbH (DE) 1998-09-16 EP disclosed