SCHEMBL7589834

SCHEMBL7589834

C=C1[C@@H](c2ccc(C(C)(C)C)cc2)[C@@](C)(c2ccc(C#N)cc2)NC(=N)N1C

nearest known ligand 0.38

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 1/20 0.38
MGAT2 Q10469 1/20 0.32
CYP3A4 P08684 1/20 0.30
HTT P42858 1/20 0.30
EPHX2 P34913 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13054165 0.87 KIF11 (0.38) KIF11MGAT2CYP3A4HTTEPHX2
SCHEMBL8195595 0.87 KIF11 (0.38) KIF11MGAT2CYP3A4HTTEPHX2
SCHEMBL7559457 0.87 KIF11 (0.38) KIF11MGAT2CYP3A4HTTEPHX2
SCHEMBL7581116 0.86 TP53 (0.31)
SCHEMBL7582435 0.82 BACE1 (0.34)
SCHEMBL7589846 0.81
SCHEMBL7581043 0.80 BACE1 (0.31)
SCHEMBL7581190 0.80 BACE1 (0.31)
SCHEMBL7584231 0.79 ELANE (0.33) CYP3A4HTT
SCHEMBL7584854 0.79 BACE1 (0.30)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8183252-B2 Heterocyclic aspartyl protease inhibitors SCHERING CORPORATION (US) 2012-05-22 US disclosed