SCHEMBL7590260

SCHEMBL7590260

O=C1CCCc2ccc(Oc3ccccc3)cc21

nearest known ligand 0.65

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MAOA P21397 12/20 0.65
MAOB P27338 12/20 0.65
CYP2A6 P11509 1/20 0.53
GSTP1 P09211 1/20 0.46
GRM5 P41594 1/20 0.44
MAPK14 Q16539 1/20 0.44
HRH3 Q9Y5N1 3/20 0.43
GPR174 Q9BXC1 1/20 0.41
PRKCI P41743 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30966021 1.00 MAOA (0.65) MAOAMAOBCYP2A6GSTP1GRM5
SCHEMBL12901556 0.87 MAOA (0.65) MAOAMAOBCYP2A6GRM5PRKCI
SCHEMBL30966017 0.87 MAOA (0.65) MAOAMAOBCYP2A6GRM5PRKCI
SCHEMBL7586081 0.84 MAOA (0.61) MAOAMAOBCYP2A6GRM5PRKCI
SCHEMBL30965992 0.82 MAOA (0.49) MAOAMAOBCYP2A6HRH3GPR174
SCHEMBL10175553 0.81 PARP10 (0.53) MAOAMAOBMAPK14
SCHEMBL21758061 0.79 HRH3 (0.62) MAOAMAOBMAPK14HRH3
SCHEMBL30067289 0.79 MAOB (1.00) MAOAMAOBGRM5
SCHEMBL3501723 0.79 MAOB (1.00) MAOAMAOBGRM5
SCHEMBL120284 0.78 MAOB (0.58) MAOAMAOBCYP2A6HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007075772-A2 COMPOUNDS, SCREENS, AND METHODS OF TREATMENT PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2007-07-05 WO disclosed
EP-0864559-B1 Substituted amino compounds and their use as analgesic active substances GRUENENTHAL GMBH (DE) 2002-06-05 EP disclosed
US-6022895-A Substituted amino compounds and their use as substances having an analgesic effect GRUENENTHAL GMBH (DE) 2000-02-08 US disclosed
EP-0864559-A1 Substituted amino compounds and their use as analgesic active substances Grünenthal GmbH (DE) 1998-09-16 EP disclosed