SCHEMBL7590349

SCHEMBL7590349

CCc1ccc(CC(=O)OC(C)(C)C)cc1N

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.49
GAA P10253 2/20 0.49
GFER P55789 1/20 0.49
MTNR1A P48039 5/20 0.47
MTNR1B P49286 5/20 0.47
RIPK1 Q13546 1/20 0.37
RIPK3 Q9Y572 1/20 0.37
SLC7A5 Q01650 2/20 0.35
TLR7 Q9NYK1 2/20 0.33
KDM4E B2RXH2 1/20 0.33
MAPT P10636 1/20 0.33
HPGD P15428 1/20 0.33
ALOX15 P16050 1/20 0.33
TSHR P16473 1/20 0.33
HSD17B10 Q99714 1/20 0.33
PPARG P37231 2/20 0.33
PPARA Q07869 1/20 0.33
RXRA P19793 1/20 0.33
NR1H2 P55055 1/20 0.33
NR1H3 Q13133 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16410352 0.91 MTNR1A (0.48) ALDH1A1GAAGFERMTNR1AMTNR1B
SCHEMBL7591321 0.85 MTNR1A (0.39) ALDH1A1GAAGFERMTNR1AMTNR1B
SCHEMBL28069959 0.85 MTNR1A (0.48) ALDH1A1GAAGFERMTNR1AMTNR1B
SCHEMBL20424475 0.84 MTNR1A (0.50) ALDH1A1GAAGFERMTNR1AMTNR1B
Hydrochloric Acid SCHEMBL7594650 0.84 MTNR1A (0.39) ALDH1A1GAAGFERMTNR1AMTNR1B
SCHEMBL28629032 0.82 ALDH1A1 (0.47) ALDH1A1GAAGFERMTNR1AMTNR1B
SCHEMBL16410349 0.82 MTNR1A (0.48) ALDH1A1GAAGFERMTNR1AMTNR1B
SCHEMBL2432439 0.81 ALDH1A1 (0.45) ALDH1A1GAAGFERMTNR1AMTNR1B
SCHEMBL5100488 0.81 ALDH1A1 (0.51) ALDH1A1GAAGFERMAPTHSD17B10
SCHEMBL23589258 0.81 MTNR1A (0.44) ALDH1A1GAAGFERMTNR1AMTNR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6368573-B1 MEASURING MYOCARDIAL FUNCTION IN MAMMAL KING PHARMACEUTICALS RESEARCH AND DEVELOPMENT, INC. 2002-04-09 US disclosed
US-5063233-A Cardiovascular disorders CIBA-GEIGY CORPORATION (US) 1991-11-05 US disclosed
US-5034381-A Antagonist CIBA-GEIGY CORPORATION (US) 1991-07-23 US disclosed
US-4968697-A ADENOSINE-2 RECEPTOR AGONISTS CIBA-GEIGY CORPORATION (US) 1990-11-06 US disclosed
US-4954504-A Hypotensive agents, psychotic disorders CIBA-GEIGY CORPORATION (US) 1990-09-04 US disclosed
EP-0323807-A2 Certain 2-substituted adenosine derivatives CIBA-GEIGY AG (CH) 1989-07-12 EP disclosed
EP-0277917-A2 Certain adenosine 5'-carboxamide derivatives CIBA-GEIGY AG (CH) 1988-08-10 EP disclosed
EP-0267878-A1 N9-cyclopentyl-substituted adenine derivatives CIBA-GEIGY AG (CH) 1988-05-18 EP disclosed