SCHEMBL7590939

SCHEMBL7590939

OB(O)Oc1ccc(C(F)(F)F)cc1C(F)(F)F

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 2/20 0.46
RXRA P19793 1/20 0.46
RXRB P28702 1/20 0.46
RXRG P48443 1/20 0.46
MGLL Q99685 2/20 0.39
TRPV6 Q9H1D0 2/20 0.39
ORAI1 Q96D31 1/20 0.39
ORAI2 Q96SN7 1/20 0.39
ORAI3 Q9BRQ5 1/20 0.39
CYP2C19 P33261 2/20 0.35
RAB9A P51151 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
KDM4E B2RXH2 1/20 0.35
USP2 O75604 1/20 0.35
ALDH1A1 P00352 1/20 0.35
HPGD P15428 1/20 0.35
HSD17B10 Q99714 1/20 0.35
PTGDR2 Q9Y5Y4 3/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2C9 P11712 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31053746 1.00 CES2 (0.46) CES2RXRARXRBRXRGMGLL
SCHEMBL28549368 0.87 CES2 (0.47) CES2RXRARXRBRXRGMGLL
SCHEMBL28949758 0.85 CES2 (0.46) CES2RXRARXRBRXRGMGLL
SCHEMBL30705412 0.81 MGLL (0.39) CES2MGLLTRPV6ORAI1ORAI2
SCHEMBL2412562 0.81 PDE2A (0.42) MGLLTRPV6ORAI1ORAI2ORAI3
SCHEMBL31351020 0.81 PDE2A (0.42) MGLLTRPV6ORAI1ORAI2ORAI3
SCHEMBL28024774 0.81 MRGPRX4 (0.43) MGLLTRPV6ORAI1ORAI2ORAI3
SCHEMBL30916840 0.80 MRGPRX4 (0.44) CYP2C19RAB9AL3MBTL1KDM4EPTGDR2
SCHEMBL2415029 0.80 MRGPRX4 (0.45)
SCHEMBL31072357 0.79 MAPT (0.43) TRPV6ORAI1ORAI2ORAI3CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0675118-B1 Biphenylderivatives, process for their preparation and their use as medicaments EISAI CO LTD (JP) 2002-10-09 EP disclosed
US-6281214-B1 USEFUL FOR TREATING AND AMELIORATING MENTAL DISORDERS EISAI CO., LTD (JP) 2001-08-28 US disclosed
EP-0675118-A2 Biphenylderivatives, process for their preparation and their use as medicaments Eisai Co., Ltd. (JP) 1995-10-04 EP disclosed