SCHEMBL7592147

SCHEMBL7592147

COc1cccc2c1CCC(CN(C)C)=C2c1cccc(O)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR7 P34969 5/20 0.45
OPRD1 P41143 2/20 0.43
ABCB1 P08183 1/20 0.39
KDM1A O60341 1/20 0.38
MAOA P21397 1/20 0.38
ADRA2A P08913 3/20 0.37
ADRA2B P18089 3/20 0.37
ADRA2C P18825 3/20 0.37
KIF11 P52732 1/20 0.37
FYN P06241 1/20 0.36
HSD11B1 P28845 2/20 0.36
HSD17B2 P37059 2/20 0.36
HSD17B1 P14061 1/20 0.36
HTR1A P08908 1/20 0.36
HTR1D P28221 1/20 0.36
HTR1B P28222 1/20 0.36
HTR2A P28223 1/20 0.36
HTR2C P28335 1/20 0.36
HTR1E P28566 1/20 0.36
HTR2B P41595 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8018161 0.99 HTR7 (0.44) HTR7OPRD1ABCB1KDM1AMAOA
SCHEMBL7591721 0.86 SLC6A4 (0.41) HTR7OPRD1ADRA2AADRA2BADRA2C
SCHEMBL7586084 0.86 HTR7 (0.50) HTR7HTR1AHTR1DHTR1BHTR2A
Hydrochloric Acid SCHEMBL8011602 0.85 SLC6A4 (0.40) HTR7OPRD1ADRA2AADRA2BADRA2C
Hydrochloric Acid SCHEMBL8002527 0.85 HTR7 (0.49) HTR7HTR1AHTR1DHTR1BHTR2A
SCHEMBL7588577 0.85 HSD17B1 (0.35) ADRA2AADRA2BADRA2CHSD17B2HSD17B1
SCHEMBL7590974 0.84 HSD17B1 (0.36) HTR7OPRD1ADRA2AADRA2BADRA2C
Hydrochloric Acid SCHEMBL8014383 0.84 HSD17B1 (0.34) ADRA2AADRA2BADRA2CHSD17B2HSD17B1
Hydrochloric Acid SCHEMBL8011897 0.83 OPRK1 (0.35) HTR7OPRD1ADRA2AADRA2BADRA2C
SCHEMBL7611357 0.82 HTR7 (0.42) HTR7OPRD1ABCB1KDM1AMAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0864559-B1 Substituted amino compounds and their use as analgesic active substances GRUENENTHAL GMBH (DE) 2002-06-05 EP disclosed
EP-0864559-A1 Substituted amino compounds and their use as analgesic active substances Grünenthal GmbH (DE) 1998-09-16 EP disclosed