SCHEMBL7596205

SCHEMBL7596205

O=C(O)c1cc(F)c(Cl)c(I)c1Cl

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 1/20 0.48
NFE2L2 Q16236 1/20 0.48
CYP3A4 P08684 1/20 0.41
MAP2K1 Q02750 1/20 0.37
KDM4E B2RXH2 1/20 0.36
ASPH Q12797 1/20 0.36
KDM8 Q8N371 1/20 0.36
ACLY P53396 1/20 0.35
TSHR P16473 2/20 0.35
ALDH1A1 P00352 1/20 0.35
TP53 P04637 1/20 0.35
CASP1 P29466 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
DAO P14920 1/20 0.35
KDM4A O75164 1/20 0.35
KDM5A P29375 1/20 0.35
KDM4C Q9H3R0 1/20 0.35
KDM5B Q9UGL1 1/20 0.35
TPMT P51580 1/20 0.34
AKR1C2 P52895 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9766052 0.84 ALDH1A1 (0.41) KEAP1NFE2L2TSHRALDH1A1
SCHEMBL8974977 0.81 KEAP1 (0.53) KEAP1NFE2L2CYP3A4KDM4EASPH
SCHEMBL26105927 0.78 KEAP1 (0.47) KEAP1NFE2L2CYP3A4MAP2K1KDM4E
SCHEMBL30574276 0.78 KEAP1 (0.47) KEAP1NFE2L2CYP3A4MAP2K1KDM4E
SCHEMBL29053402 0.78 KDM4E (0.47) KEAP1NFE2L2CYP3A4KDM4ETPMT
SCHEMBL8038276 0.76 KEAP1 (0.48) KEAP1NFE2L2CYP3A4KDM4EASPH
SCHEMBL7041352 0.76 CYP3A4 (0.50) KEAP1NFE2L2CYP3A4KDM4EASPH
SCHEMBL10539386 0.76 KEAP1 (0.48) KEAP1NFE2L2CYP3A4KDM4EASPH
SCHEMBL22972614 0.75 KEAP1 (0.52) KEAP1NFE2L2CYP3A4MAP2K1KDM4E
SCHEMBL3539441 0.75 KEAP1 (0.52) KEAP1NFE2L2CYP3A4MAP2K1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0968994-B1 PROCESS FOR PRODUCING SUBSTITUTED TRIFLUOROBENZOIC ACIDS AND ESTERS THEREOF UBE INDUSTRIES (JP) 2002-11-06 EP disclosed
US-6307091-B1 TRIFLUOROMETHYLATING A TRIFLUOROIODOBENZOIC ACID ESTER WITH ADIFLUORO(FLUOROSULFONYL)ACETIC ACID ESTER IN THE PRESENCE OF A COPPER CATALYST IN AN ORGANIC SOLVENT. UBE INDUSTRIES, LTD. (JP) 2001-10-23 US disclosed
US-6160171-A Trifluoro-substituted benzoic acid, esters thereof, and process for producing the same UBE INDUSTRIES, LTD. (JP) 2000-12-12 US disclosed
EP-0968994-A1 SUBSTITUTED TRIFLUOROBENZOIC ACIDS, ESTERS THEREOF, AND PROCESS FOR PRODUCING THE SAME UBE INDUSTRIES, LTD. (JP) 2000-01-05 EP disclosed
EP-0266512-B1 METHOD FOR THE PRODUCTION OF BENZOIC ACID DERIVATIVES FLUORINATED ON THE NUCLEUS BAYER AG (DE) 1991-12-04 EP disclosed
US-4990661-A Process for the preparation of benzoic acid derivatives BAYER AKTIENGESELLSCHAFT (DE) 1991-02-05 US disclosed
US-4851160-A Process for the preparation of benzoic acid derivatives BAYER AKTIENGESELLSCHAFT (DE) 1989-07-25 US disclosed
EP-0266512-A2 Method for the production of benzoic acid derivatives fluorinated on the nucleus BAYER AG (DE) 1988-05-11 EP disclosed