SCHEMBL7596705

SCHEMBL7596705

NC(=S)Nc1ccc(CCN2CCc3ccccc3C2)cc1

nearest known ligand 0.65

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 11/20 0.65
ABCG2 Q9UNQ0 9/20 0.65
DRD2 P14416 1/20 0.62
TNF P01375 1/20 0.57
NOD1 Q9Y239 1/20 0.57
ALOX15 P16050 2/20 0.53
MEN1 O00255 1/20 0.53
TP53 P04637 1/20 0.53
KMT2A Q03164 1/20 0.53
KDM4E B2RXH2 1/20 0.52
CYP1A2 P05177 1/20 0.51
CYP3A4 P08684 1/20 0.51
CYP2D6 P10635 1/20 0.51
CYP2C19 P33261 1/20 0.51
MAPT P10636 1/20 0.51
USP2 O75604 1/20 0.50
TAAR1 Q96RJ0 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7597148 0.82 ABCB1 (0.62) ABCB1ABCG2DRD2TNFNOD1
SCHEMBL4047473 0.82 ABCB1 (0.80) ABCB1ABCG2DRD2TNFNOD1
SCHEMBL4047475 0.79 ABCB1 (1.00) ABCB1ABCG2DRD2TNFNOD1
SCHEMBL24349700 0.78 ABCB1 (0.70) ABCB1ABCG2DRD2KDM4E
SCHEMBL7595478 0.78 ABCB1 (0.61) ABCB1ABCG2DRD2TNFNOD1
SCHEMBL6512477 0.78 HRH3 (0.68) DRD2KDM4E
Hydrochloric Acid SCHEMBL7600991 0.77 ABCB1 (0.68) ABCB1ABCG2DRD2
SCHEMBL3429411 0.75 EED (0.51) MEN1TP53KMT2AMAPTTAAR1
SCHEMBL16061507 0.74 ABCB1 (0.64) ABCB1ABCG2DRD2TNFNOD1
SCHEMBL8491977 0.72 DRD2 (0.59) ABCB1ABCG2DRD2TNFNOD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0782567-B2 ISOTHIOUREA DERIVATIVES AS NO SYNTHASE INHIBITORS ASTRA AB (SE) 2002-12-11 EP disclosed
EP-0782567-B1 ISOTHIOUREA DERIVATIVES AS NO SYNTHASE INHIBITORS ASTRA AB (SE) 1999-06-30 EP disclosed