SCHEMBL7597587

SCHEMBL7597587

COC(=O)C1CCc2ccsc2C1N(C(=O)OC)c1ccccc1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 2/20 0.37
ALDH1A1 P00352 1/20 0.37
MAPT P10636 1/20 0.37
HPGD P15428 1/20 0.37
ALOX15 P16050 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
KMT2A Q03164 1/20 0.34
OPRM1 P35372 3/20 0.34
GRIN2B Q13224 5/20 0.33
SLC6A4 P31645 4/20 0.33
SLC6A2 P23975 3/20 0.33
SLC6A3 Q01959 2/20 0.33
CYP3A4 P08684 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2D6 P10635 1/20 0.33
TSHR P16473 1/20 0.33
MAPK1 P28482 1/20 0.33
CHRM4 P08173 1/20 0.33
CHRM5 P08912 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7596481 0.91 SLC6A4 (0.36) HSD17B10ALDH1A1MAPTKMT2AOPRM1
SCHEMBL7597646 0.75 ALDH1A1 (0.38) HSD17B10ALDH1A1MAPTHPGDALOX15
SCHEMBL7609208 0.74 KMT2A (0.43) KMT2ASLC6A4SLC6A2SLC6A3
SCHEMBL7596854 0.72 ALDH1A1 (0.36) HSD17B10ALDH1A1MAPTHPGDNPSR1
SCHEMBL7593413 0.70 ALDH1A1 (0.41) HSD17B10ALDH1A1MAPTHPGDALOX15
SCHEMBL28660867 0.64 ALDH1A1 (0.42) HSD17B10ALDH1A1MAPTHPGDALOX15
SCHEMBL28249129 0.64 ALDH1A1 (0.59) HSD17B10ALDH1A1MAPTHPGDALOX15
SCHEMBL28768033 0.62 OPRM1 (0.49) HSD17B10ALDH1A1MAPTHPGDALOX15
SCHEMBL7613074 0.62 KMT2A (0.56) ALDH1A1MAPTKMT2AOPRM1GRIN2B
SCHEMBL10581361 0.61 PIN1 (0.46) HSD17B10MAPTKMT2ASLC6A4CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0690054-B1 1-Amino-2-cyclohexene derivatives and production process therefor KURARAY CO (JP) 2002-11-20 EP disclosed
US-5587486-A CONDENSATION; CARBONYLATION; HYDROLYSIS; INTERMEDIATES IN THE PRODUCTION OF MEDICINAL AND AGRICULTURAL AGENTS KURARAY CO., LTD. (JP) 1996-12-24 US disclosed
EP-0690054-A1 1-Amino-2-cyclohexene derivatives and production process therefor KURARAY CO., LTD. (JP) 1996-01-03 EP disclosed