SCHEMBL7598202

SCHEMBL7598202

CCCCOC(=O)N[C@@H](C)C(=O)NC1C(=O)N(c2ccccc2)c2ccccc2N(c2ccccc2)C1=O

nearest known ligand 0.53

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CCKBR P32239 14/20 0.53
XIAP P98170 4/20 0.47
CCKAR P32238 7/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7849872 0.89 PSEN1 (0.48) CCKBRXIAP
SCHEMBL6920745 0.82 CCKBR (0.41) CCKBRXIAP
SCHEMBL4411787 0.81 XIAP (0.48) CCKBRXIAPCCKAR
SCHEMBL4417220 0.74 PSEN1 (0.59) CCKBRXIAPCCKAR
SCHEMBL7847907 0.74 CCKBR (0.54) CCKBRXIAPCCKAR
SCHEMBL4424536 0.74 XIAP (0.49) CCKBRXIAPCCKAR
SCHEMBL4417467 0.73 PSEN1 (0.68)
SCHEMBL6301491 0.71 CCKBR (0.50) CCKBRXIAPCCKAR
SCHEMBL8020336 0.70 ALDH1A1 (0.52) CCKBRXIAP
SCHEMBL17164501 0.70 CTSK (0.49)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0951466-A2 CYCLOALKYL, LACTAM, LACTONE AND RELATED COMPOUNDS, PHARMACEUTICAL COMPOSITIONS COMPRISING SAME, AND METHODS FOR INHIBITING BETA-AMYLOID PEPTIDE RELEASE AND/OR ITS SYNTHESIS BY USE OF SUCH COMPOUNDS Elan Pharmaceuticals, Inc. (US) 1999-10-27 EP disclosed
WO-1998028268-A2 CYCLOALKYL, LACTAM, LACTONE AND RELATED COMPOUNDS AS β-AMYLOID PEPTIDE RELEASE INHIBITORS ELAN PHARMACEUTICALS, INC. (US) 1998-07-02 WO disclosed