SCHEMBL7599437

SCHEMBL7599437

CC[C@H](C)[C@H](NC(=O)OCC1c2ccccc2-c2ccccc21)C(=O)OC[C@@H](OC(=O)[C@@H](NC(=O)OCC1c2ccccc2-c2ccccc21)[C@@H](C)CC)C(=O)O

nearest known ligand 0.47

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CASP3 P42574 4/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2D6 P10635 1/20 0.46
CYP2C9 P11712 1/20 0.46
CYP2C19 P33261 1/20 0.46
RAB9A P51151 1/20 0.46
MDM4 O15151 2/20 0.43
TP53 P04637 2/20 0.43
PIN1 Q13526 1/20 0.43
TLR2 O60603 2/20 0.42
KMT2A Q03164 2/20 0.42
MDM2 Q00987 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7599890 0.91 CASP3 (0.52) CASP3MDM4TP53PIN1TLR2
SCHEMBL8132183 0.88 CASP3 (0.48) CASP3CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL1486214 0.86 CASP3 (0.52) CASP3CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL118209 0.86 CASP3 (0.52) CASP3CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL1486287 0.86 CASP3 (0.52) CASP3CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL6038102 0.86 CASP3 (0.52) CASP3CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL1564185 0.86 CASP3 (0.52) CASP3CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL119497 0.86 CASP3 (0.52) CASP3CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL30896049 0.86 CASP3 (0.52) CASP3CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL30896048 0.86 CASP3 (0.52) CASP3CYP3A4CYP2D6CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2002503673-A 2002-02-05 JP claimed
EP-1054891-A1 PRODRUGS MEDIVIR AB (SE) 2000-11-29 EP claimed
WO-1999041275-A1 PRODRUGS MEDIVIR AB (SE) 1999-08-19 WO claimed