Isatin

Isatin

SCHEMBL76012

O=C1Nc2ccccc2C1=O.Oc1ccccc1.Oc1ccccc1

nearest known ligand 0.77

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 10/20 0.77
MAOB P27338 10/20 0.77
PLK4 O00444 2/20 0.54
PLK1 P53350 2/20 0.54
RET P07949 1/20 0.54
FLT3 P36888 1/20 0.54
PDGFRB P09619 1/20 0.54
LRRK2 Q5S007 2/20 0.53
PDGFRA P16234 1/20 0.53
FER P16591 1/20 0.53
LTK P29376 1/20 0.53
CDK8 P49336 1/20 0.53
ACVR1 Q04771 1/20 0.53
DYRK1B Q9Y463 1/20 0.53
MAPT P10636 3/20 0.51
MEN1 O00255 2/20 0.51
ALDH1A1 P00352 2/20 0.51
KMT2A Q03164 2/20 0.51
NPSR1 Q6W5P4 2/20 0.51
LMNA P02545 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Isatin SCHEMBL28142968 1.00 MAOA (0.77) MAOAMAOBPLK4PLK1RET
Isatin SCHEMBL28365971 0.90 MAOA (0.95) MAOAMAOBFLT3LRRK2PDGFRA
Tannin Pyrogallol SCHEMBL29283471 0.90 MAOA (0.67) MAOAMAOBPLK4PLK1RET
Isatin SCHEMBL13725994 0.88 MAOA (0.83) MAOAMAOBLRRK2PDGFRAFER
Isatin SCHEMBL34016 0.88 MAOA (1.00) MAOAMAOBLRRK2PDGFRAFER
Isatin SCHEMBL973760 0.88 MAOA (1.00) MAOAMAOBLRRK2PDGFRAFER
Isatin SCHEMBL27858156 0.86 MAOA (0.87) MAOAMAOBLRRK2PDGFRAFER
Isatin SCHEMBL23256320 0.86 MAOA (0.95) MAOAMAOBLRRK2PDGFRAFER
Isatin SCHEMBL4092377 0.86 MAOA (0.95) MAOAMAOBLRRK2PDGFRAFER
Isatin SCHEMBL11646710 0.86 MAOA (0.95) MAOAMAOBLRRK2PDGFRAFER

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 3093 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4263708-B1 FIRE RETARDANT POLYCARBONATE COMPOSITIONS FOR TRANSPARENT THIN-WALL APPLICATIONS SHPP GLOBAL TECH BV (NL) 2024-04-10 EP claimed
US-20240010832-A1 FIRE RETARDANT POLYCARBONATE COMPOSITIONS FOR TRANSPARENT THIN-WALL APPLICATIONS SHPP GLOBAL TECHNOLOGIES B.V. (NL) 2024-01-11 US claimed
EP-4263708-A1 FIRE RETARDANT POLYCARBONATE COMPOSITIONS FOR TRANSPARENT THIN-WALL APPLICATIONS SHPP Global Technologies B.V. (NL) 2023-10-25 EP claimed
WO-2022130211-A1 FIRE RETARDANT POLYCARBONATE COMPOSITIONS FOR TRANSPARENT THIN‑WALL APPLICATIONS SHPP GLOBAL TECHNOLOGIES B.V. (NL) 2022-06-23 WO claimed
EP-2670798-B1 COLOR AND HEAT STABLE POLYCARBONATE COMPOSITIONS AND METHODS OF MAKING SABIC GLOBAL TECHNOLOGIES BV (NL) 2020-11-04 EP claimed
CN-111793341-A Branched high heat polycarbonate, method of manufacture and articles thereof 沙特基础工业全球技术有限公司 2020-10-20 CN claimed
EP-3719066-A1 BRANCHED, HIGH HEAT POLYCARBONATES, METHODS OF MANUFACTURE, AND ARTICLES PREPARED THEREFROM SABIC Global Technologies B.V. (NL) 2020-10-07 EP claimed
US-20200308398-A1 BRANCHED, HIGH HEAT POLYCARBONATES, METHODS OF MANUFACTURE, AND ARTICLES PREPARED THEREFROM SHPP GLOBAL TECHNOLOGIES B.V. (NL) 2020-10-01 US claimed
CN-104684973-B Fire-retardant polycarbonate film 沙特基础全球技术有限公司 2017-08-04 CN claimed
US-9580595-B2 Compositions and articles of manufacture containing branched polycarbonate SABIC GLOBAL TECHNOLOGIES B.V. (NL) 2017-02-28 US claimed
EP-1412430-B1 TRANSPARENT, FIRE-RESISTANT POLYCARBONATE COMPOSITIONS GEN ELECTRIC (US) 2008-09-03 EP claimed
WO-2008060714-A2 THERMOPLASTIC COMPOSITIONS, METHODS OF MAKING, AND ARTICLES FORMED THEREFROM SABIC INNOVATIVE PLASTICS IP B.V. (NL) 2008-05-22 WO claimed
WO-2008061140-A1 THERMOPLASTIC COMPOSITION, METHOD OF MAKING, AND ARTICLES FORMED THEREFROM SABIC INNOVATIVE PLASTICS IP BV (US) 2008-05-22 WO claimed
US-20080119631-A1 THERMOPLASTIC COMPOSITION, METHOD OF MAKING, AND ARTICLES FORMED THEREFROM GENERAL ELECTRIC COMPANY (US) 2008-05-22 US claimed
US-20080081855-A1 THERMOPLASTIC COMPOSITIONS, METHODS OF MAKING, AND ARTICLES FORMED THEREFROM GENERAL ELECTRIC COMPANY (US) 2008-04-03 US claimed
EP-1412430-A1 TRANSPARENT, FIRE-RESISTANT POLYCARBONATE COMPOSITIONS GENERAL ELECTRIC COMPANY (US) 2004-04-28 EP claimed
US-20030027905-A1 Transparent, fire-resistant polycarbonate compositions GENERAL ELECTRIC COMPANY 2003-02-06 US claimed
WO-2003008501-A1 TRANSPARENT, FIRE-RESISTANT POLYCARBONATE COMPOSITIONS GENERAL ELECTRIC COMPANY (US) 2003-01-30 WO claimed
US-5441997-A Comprising fillers, stabilizers of phosphites, phosphates and styrene-rubber impact modifier GENERAL ELECTRIC COMPANY (US) 1995-08-15 US claimed
US-5021541-A Better flowability and moblability MITSUBISHI GAS CHEMICAL CO., LTD. (JP) 1991-06-04 US claimed