SCHEMBL7601350

SCHEMBL7601350

CCN1CCNCC1Oc1ccccc1C(F)(F)F

nearest known ligand 0.42

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 7/20 0.42
HTR2A P28223 5/20 0.42
KCNH2 Q12809 1/20 0.42
SLC6A2 P23975 2/20 0.37
SLC6A4 P31645 2/20 0.37
SLC6A3 Q01959 2/20 0.37
HTR1A P08908 1/20 0.37
SSTR4 P31391 1/20 0.37
HTR2B P41595 4/20 0.37
SCD O00767 3/20 0.37
MITF O75030 1/20 0.36
DRD2 P14416 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14833412 0.81 KDM4E (0.41) HTR2ASSTR4SCD
SCHEMBL27889106 0.77 HRH1 (0.40) HTR2CKCNH2SLC6A2SLC6A4SLC6A3
SCHEMBL6446140 0.75 HTR2C (0.50) HTR2CHTR2AHTR2B
SCHEMBL2819314 0.70 HTR1A (0.58) HTR2CSLC6A2SLC6A4SLC6A3HTR1A
SCHEMBL1782071 0.70 HTR1A (0.58) HTR2CSLC6A2SLC6A4SLC6A3HTR1A
SCHEMBL7888184 0.70 HTR1A (0.58) HTR2CSLC6A2SLC6A4SLC6A3HTR1A
SCHEMBL22462919 0.69 LTA4H (0.46) HTR1ASSTR4SCDDRD2
Hydrochloric Acid SCHEMBL2947998 0.69 HTR1A (0.57) HTR2CSLC6A2SLC6A4SLC6A3HTR1A
SCHEMBL1230447 0.69 SLC6A2 (0.54) HTR2CSLC6A2SLC6A4SLC6A3HTR1A
SCHEMBL6255525 0.69 SIGMAR1 (0.43) HTR2CHTR2AKCNH2SLC6A2SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1246820-A1 NOVEL HETEROARYL DERIVATIVES, THEIR PREPARATION AND USE H. LUNDBECK A/S (DK) 2002-10-09 EP disclosed
WO-2001049683-A1 NOVEL HETEROARYL DERIVATIVES, THEIR PREPARATION AND USE H. LUNDBECK A/S (DK) 2001-07-12 WO disclosed