SCHEMBL7601554

SCHEMBL7601554

CN(c1ccccc1)S(=O)(=O)c1ccc2c(c1)C(=O)C(=O)N2

nearest known ligand 0.58

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CASP3 P42574 9/20 0.58
MAOA P21397 5/20 0.58
CA12 O43570 2/20 0.55
CA9 Q16790 2/20 0.55
MAOB P27338 4/20 0.54
CA1 P00915 1/20 0.54
CA2 P00918 1/20 0.54
CASP7 P55210 2/20 0.52
CASP2 P42575 1/20 0.52
CASP6 P55212 1/20 0.52
POLB P06746 1/20 0.51
HTR2C P28335 1/20 0.50
HTR2B P41595 1/20 0.50
ATM Q13315 1/20 0.49
L3MBTL1 Q9Y468 1/20 0.49
CASP1 P29466 1/20 0.48
CASP9 P55211 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4411083 0.82 CASP3 (0.64) CASP3MAOACA12CA9MAOB
SCHEMBL4906814 0.80 MAOA (0.78) CASP3MAOACA12CA9MAOB
SCHEMBL20302942 0.79 CA12 (0.60) CA12CA9POLBHTR2CHTR2B
SCHEMBL6536379 0.78 CASP3 (0.78) CASP3CASP7CASP2CASP6CASP1
SCHEMBL6535436 0.78 CASP3 (0.67) CASP3MAOACA12CA9MAOB
SCHEMBL3248876 0.76 ALDH1A1 (0.62) CA12CA9POLBHTR2CHTR2B
SCHEMBL7566978 0.75 CASP3 (0.74) CASP3MAOACA12CA9MAOB
SCHEMBL5893648 0.74 CA12 (0.69) CASP3MAOACA12CA9MAOB
SCHEMBL6535335 0.72 CASP3 (1.00) CASP3MAOACA12CA9MAOB
SCHEMBL3822617 0.72 CA12 (1.00) CA12CA9ATML3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6403792-B1 INHIBIT PRODUCTION OF CASPASE 3 AND 7 IN MAMMALS SMITHKLINE BEECHAM CORPORATION 2002-06-11 US claimed
EP-1001933-A4 CASPASES AND APOPTOSIS SMITHKLINE BEECHAM CORP (US) 2002-11-06 EP disclosed
US-6403792-B1 INHIBIT PRODUCTION OF CASPASE 3 AND 7 IN MAMMALS SMITHKLINE BEECHAM CORPORATION 2002-06-11 US disclosed
EP-1001933-A1 CASPASES AND APOPTOSIS SMITHKLINE BEECHAM CORPORATION (US) 2000-05-24 EP disclosed
WO-1999006367-A1 CASPASES AND APOPTOSIS SMITHKLINE BEECHAM CORPORATION (US) 1999-02-11 WO disclosed