SCHEMBL7601597

SCHEMBL7601597

COc1cccc(OCCOc2nccnc2N2CCNCC2)c1.OCCOc1cccc(OCCOc2nccnc2N2CCNCC2)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB1 P08588 2/20 0.47
CYP1A2 P05177 2/20 0.47
CYP3A4 P08684 2/20 0.47
USP2 O75604 1/20 0.47
CYP2C19 P33261 1/20 0.47
HSD17B10 Q99714 1/20 0.47
CLK4 Q9HAZ1 1/20 0.47
HTR6 P50406 4/20 0.45
TSHR P16473 2/20 0.44
TP53 P04637 1/20 0.44
CYP2D6 P10635 1/20 0.44
HTR1A P08908 2/20 0.43
HTR7 P34969 2/20 0.43
HTR2B P41595 2/20 0.43
HTR3A P46098 2/20 0.43
HTR2A P28223 1/20 0.43
HTR2C P28335 1/20 0.43
TGFBR1 P36897 1/20 0.42
ACVR1 Q04771 1/20 0.42
ALDH1A1 P00352 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4313451 0.94 KDM4E (0.39) ADRB1CYP1A2CYP3A4USP2CYP2C19
SCHEMBL4315672 0.94 ADRB1 (0.52) ADRB1CYP1A2CYP3A4USP2CYP2C19
SCHEMBL7476206 0.91 ADRB1 (0.51) ADRB1CYP1A2CYP3A4USP2CYP2C19
SCHEMBL2640084 0.88 CHRNB2 (0.49) ADRB1CYP1A2CYP3A4USP2CYP2C19
SCHEMBL4308724 0.85 EPHX2 (0.40) ADRB1HTR6HTR1AHTR2C
SCHEMBL4326917 0.85 HTR2C (0.39) HTR2C
SCHEMBL4309052 0.85 ADRB1 (0.50) ADRB1CYP1A2CYP3A4USP2CYP2C19
SCHEMBL4312805 0.85 HTR6 (0.48) ADRB1CYP1A2CYP3A4USP2CYP2C19
SCHEMBL4320133 0.84 HTR2C (0.42) ADRB1CYP1A2CYP3A4USP2CYP2C19
SCHEMBL4324680 0.84 HTR6 (0.39) HTR6HTR2CALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1178973-A2 NOVEL COMPOUNDS, THEIR USE AND PREPARATION Pharmacia AB (SE) 2002-02-13 EP disclosed
WO-2000076984-A2 NOVEL COMPOUNDS, THEIR USE AND PREPARATION BIOVITRUM AB (SE) 2000-12-21 WO disclosed