SCHEMBL7601654

SCHEMBL7601654

Cc1ccc(C#N)cc1[C@@]1(C)NC(=N)N(C)C(=O)[C@@H]1c1ccc(C(C)(F)F)cc1

nearest known ligand 0.33

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ELANE P08246 11/20 0.33
CYP2C9 P11712 3/20 0.33
P2RX7 Q99572 2/20 0.31
CYP3A4 P08684 2/20 0.31
HTR7 P34969 1/20 0.31
FASN P49327 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13081547 1.00 ELANE (0.33) ELANECYP2C9P2RX7CYP3A4HTR7
SCHEMBL7552777 0.91 HSD11B1 (0.32) ELANE
SCHEMBL13054185 0.91 HSD11B1 (0.32) ELANE
SCHEMBL8210521 0.85 BACE1 (0.35) ELANECYP2C9CYP3A4
SCHEMBL7547187 0.85 BACE1 (0.35) ELANECYP2C9CYP3A4
SCHEMBL13081258 0.84 TDP1 (0.31)
SCHEMBL8412215 0.82 PGR (0.33)
SCHEMBL7560896 0.82 ELANE (0.31) ELANE
SCHEMBL13053899 0.82 ELANE (0.31) ELANE
SCHEMBL7546301 0.82 HTR7 (0.31) HTR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8183252-B2 Heterocyclic aspartyl protease inhibitors SCHERING CORPORATION (US) 2012-05-22 US disclosed