SCHEMBL7602580

SCHEMBL7602580

COc1ncccc1C(N)CCCOc1cc(Cl)ccc1C#N

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 9/20 0.40
SLC6A2 P23975 9/20 0.40
SLC6A4 P31645 9/20 0.40
NOS2 P35228 8/20 0.40
KCNH2 Q12809 2/20 0.38
SCN9A Q15858 1/20 0.37
SLC22A12 Q96S37 3/20 0.36
NPC1 O15118 2/20 0.36
RAB9A P51151 2/20 0.36
KDM4E B2RXH2 1/20 0.36
MAPT P10636 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
CYP3A4 P08684 3/20 0.34
SLC6A3 Q01959 2/20 0.34
F11 P03951 1/20 0.34
AR P10275 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6575059 0.80 NOS2 (0.53) CYP2D6SLC6A2SLC6A4NOS2KCNH2
Oxalic Acid SCHEMBL6576500 0.76 NOS2 (0.58) CYP2D6SLC6A2SLC6A4NOS2KCNH2
SCHEMBL7604472 0.71 NOS2 (0.43) CYP2D6SLC6A2SLC6A4NOS2KCNH2
SCHEMBL7608216 0.70 NOS2 (0.42) CYP2D6SLC6A2SLC6A4NOS2KCNH2
SCHEMBL4678021 0.68 KDM4E (0.54) CYP2D6SLC6A2SLC6A4NOS2KCNH2
SCHEMBL7604530 0.67 NOS2 (0.43) CYP2D6SLC6A2SLC6A4NOS2KCNH2
SCHEMBL4857820 0.66 AR (0.53) CYP2D6SLC6A2SLC6A4NOS2KDM4E
SCHEMBL7608154 0.65 CYP2D6 (0.40) CYP2D6SLC6A2SLC6A4NOS2KCNH2
SCHEMBL1306764 0.65 IDH1 (0.53) CYP2D6SLC6A2SLC6A4NOS2KCNH2
SCHEMBL22445567 0.64 FAAH (0.44) CYP2D6SLC6A2SLC6A4NPC1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1263714-A1 NOVEL PHENYLHETEROALKYLAMINE DERIVATIVES AstraZeneca AB (SE) 2002-12-11 EP disclosed
WO-2001062713-A1 NOVEL PHENYLHETEROALKYLAMINE DERIVATIVES ASTRAZENECA AB (SE) 2001-08-30 WO disclosed