SCHEMBL7604530

SCHEMBL7604530

N#Cc1ccc(Cl)cc1OCCC(N)c1ccc(Br)nc1

nearest known ligand 0.43

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NOS2 P35228 9/20 0.43
CYP2D6 P10635 7/20 0.43
SLC6A2 P23975 7/20 0.43
SLC6A4 P31645 7/20 0.43
KCNH2 Q12809 2/20 0.39
S1PR3 Q99500 7/20 0.36
S1PR1 P21453 5/20 0.36
S1PR4 O95977 2/20 0.36
S1PR2 O95136 2/20 0.35
SLC22A12 Q96S37 1/20 0.34
TRPV4 Q9HBA0 1/20 0.34
P2RX3 P56373 1/20 0.34
P2RX2 Q9UBL9 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6490535 0.80 NOS2 (0.67) NOS2CYP2D6SLC6A2SLC6A4KCNH2
Oxalic Acid SCHEMBL6501478 0.75 NOS2 (0.71) NOS2CYP2D6SLC6A2SLC6A4KCNH2
SCHEMBL7608216 0.74 NOS2 (0.42) NOS2CYP2D6SLC6A2SLC6A4KCNH2
SCHEMBL7604472 0.73 NOS2 (0.43) NOS2CYP2D6SLC6A2SLC6A4KCNH2
SCHEMBL1306764 0.69 IDH1 (0.53) NOS2CYP2D6SLC6A2SLC6A4KCNH2
SCHEMBL6981893 0.68 NOS2 (0.52) NOS2CYP2D6SLC6A2SLC6A4KCNH2
SCHEMBL7602580 0.67 CYP2D6 (0.40) NOS2CYP2D6SLC6A2SLC6A4KCNH2
SCHEMBL7604665 0.67 NOS2 (0.39) NOS2CYP2D6SLC6A2SLC6A4KCNH2
SCHEMBL4678021 0.66 KDM4E (0.54) NOS2CYP2D6SLC6A2SLC6A4KCNH2
SCHEMBL13358872 0.66 SLC2A1 (0.37) SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1263711-A1 NOVEL USE OF PHENYLHETEROALKYLAMINE DERIVATIVES AstraZeneca AB (SE) 2002-12-11 EP disclosed
WO-2001062704-A1 NOVEL USE OF PHENYLHETEROALKYLAMINE DERIVATIVES ASTRAZENECA AB (SE) 2001-08-30 WO disclosed