SCHEMBL7604066

SCHEMBL7604066

COc1ccc2c(c1)C(C)(C)CC=C2

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 7/20 0.40
CA12 O43570 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
CA7 P43166 1/20 0.38
CA9 Q16790 1/20 0.38
CA14 Q9ULX7 1/20 0.38
GAA P10253 1/20 0.36
HTR2C P28335 1/20 0.35
EHMT2 Q96KQ7 1/20 0.35
ALDH1A1 P00352 2/20 0.34
MAPT P10636 2/20 0.34
CYP3A4 P08684 1/20 0.34
MEN1 O00255 1/20 0.34
THRB P10828 1/20 0.34
KMT2A Q03164 1/20 0.34
MAOA P21397 1/20 0.34
MAOB P27338 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28239399 0.88 CA12 (0.39) CA12CA1CA2CA7CA9
SCHEMBL7601929 0.82 PDK2 (0.37) SIGMAR1CA12CA9GAAALDH1A1
SCHEMBL7603353 0.75 NPC1 (0.46) MAOAMAOB
SCHEMBL30659806 0.75 AKR1B1 (0.33) HTR2C
SCHEMBL15266966 0.72 CA12 (0.35) CA12CA1CA2CA7CA9
SCHEMBL869051 0.70 IDO1 (0.34)
SCHEMBL4420031 0.70 RXRA (0.53) CA12CA1CA2CA7CA9
SCHEMBL4369386 0.70 HIF1A (0.33) GAAMAPTMAOA
SCHEMBL30320303 0.70 HIF1A (0.33) GAAMAPTMAOA
SCHEMBL10533866 0.70 CA1 (0.42) CA12CA1CA2CA7CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1265848-A2 AMINES SUBSTITUTED WITH A DIHYDRONAPHTHALENYL, CRHOMENYL, OR THIOCHROMENYL GROUP, AN ARYL OR HETEROARYL GROUP AND AN ALKYL GROUP, HAVING RETINOID-LIKE BIOLOGICAL ACTIVITY Allergan Sales, Inc. (US) 2002-12-18 EP disclosed
WO-2001070668-A2 AMINES SUBSTITUTED WITH A DIHYDRONAPHTHALENYL, CRHOMENYL, OR THIOCHROMENYL GROUP, AN ARYL OR HETEROARYL GROUP AND AN ALKYL GROUP, HAVING RETINOID-LIKE BIOLOGICAL ACTIVITY ALLERGAN, INC. (US) 2001-09-27 WO disclosed