SCHEMBL7601929

SCHEMBL7601929

CC(C)Oc1ccc2c(c1)C(C)(C)CC=C2

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDK2 Q15119 1/20 0.37
ALDH1A1 P00352 3/20 0.36
KMT2A Q03164 2/20 0.34
PARP10 Q53GL7 1/20 0.33
BRD4 O60885 1/20 0.33
BRPF1 P55201 1/20 0.33
GRIN2D O15399 1/20 0.33
GRIN3B O60391 1/20 0.33
GRIN1 Q05586 1/20 0.33
GRIN2A Q12879 1/20 0.33
GRIN2B Q13224 1/20 0.33
GRIN2C Q14957 1/20 0.33
GRIN3A Q8TCU5 1/20 0.33
HIF1A Q16665 1/20 0.32
EPAS1 Q99814 1/20 0.32
POLB P06746 1/20 0.32
ALDH1A3 P47895 1/20 0.32
ABL1 P00519 1/20 0.32
GLA P06280 1/20 0.31
KDM4E B2RXH2 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7604066 0.82 SIGMAR1 (0.40) ALDH1A1KMT2ASIGMAR1CA12CA9
SCHEMBL7610066 0.76 MAOA (0.41) PDK2ALDH1A1KMT2AKDM4EHPGD
SCHEMBL7629290 0.72 OPRD1 (0.34) ALDH1A1HIF1AEPAS1ABL1HSD17B10
SCHEMBL7603353 0.72 NPC1 (0.46) PARP10HPGD
SCHEMBL30659806 0.71 AKR1B1 (0.33) HIF1AEPAS1
SCHEMBL30218170 0.70 ALDH1A1 (0.40) PDK2ALDH1A1KMT2APARP10BRD4
SCHEMBL30218032 0.70 ALDH1A1 (0.40) ALDH1A1KMT2APARP10BRD4BRPF1
SCHEMBL8170079 0.70 HIF1A (0.33) HIF1AEPAS1
SCHEMBL10828062 0.67 TLK2 (0.38) PDK2ALDH1A1KMT2APARP10BRD4
SCHEMBL4369386 0.66 HIF1A (0.33) HIF1AEPAS1KDM4EGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1265848-A2 AMINES SUBSTITUTED WITH A DIHYDRONAPHTHALENYL, CRHOMENYL, OR THIOCHROMENYL GROUP, AN ARYL OR HETEROARYL GROUP AND AN ALKYL GROUP, HAVING RETINOID-LIKE BIOLOGICAL ACTIVITY Allergan Sales, Inc. (US) 2002-12-18 EP disclosed
WO-2001070668-A2 AMINES SUBSTITUTED WITH A DIHYDRONAPHTHALENYL, CRHOMENYL, OR THIOCHROMENYL GROUP, AN ARYL OR HETEROARYL GROUP AND AN ALKYL GROUP, HAVING RETINOID-LIKE BIOLOGICAL ACTIVITY ALLERGAN, INC. (US) 2001-09-27 WO disclosed