SCHEMBL7605286

SCHEMBL7605286

Nc1cc([C@@H](O)CN(CCC(c2ccc(N3CCCC3)cc2)c2ccc(N3CCCC3)cc2)Cc2ccccc2)ccc1OCc1ccccc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
KDM4E B2RXH2 2/20 0.39
ALDH1A1 P00352 2/20 0.39
GAA P10253 2/20 0.39
MAPT P10636 2/20 0.39
TP53 P04637 1/20 0.39
ALOX12 P18054 1/20 0.39
MAPK1 P28482 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
LRRK2 Q5S007 2/20 0.36
DPP7 Q9UHL4 1/20 0.36
RORC P51449 2/20 0.36
CNR2 P34972 2/20 0.34
GRIN1 Q05586 1/20 0.34
GRIN2B Q13224 1/20 0.34
HTR6 P50406 2/20 0.34
ADRA1D P25100 2/20 0.34
ADRA1A P35348 2/20 0.34
ADRA1B P35368 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7608453 0.86 ALOX5 (0.40) MEN1KMT2AALDH1A1GAAMAPT
SCHEMBL7604462 0.86 POLB (0.46) MEN1KMT2AKDM4EALDH1A1GAA
SCHEMBL7685567 0.84 ADRB3 (0.43) MEN1KMT2AKDM4EALDH1A1GAA
SCHEMBL7685564 0.84 ADRB3 (0.43) MEN1KMT2AKDM4EALDH1A1GAA
SCHEMBL7607631 0.84 NR1H3 (0.44) MEN1KMT2AALDH1A1MAPTTP53
SCHEMBL7607627 0.84 NR1H3 (0.44) MEN1KMT2AALDH1A1MAPTTP53
SCHEMBL7605293 0.82 KDM4E (0.39) MEN1KMT2AKDM4EALDH1A1GAA
SCHEMBL11670452 0.81 MEN1 (0.39) MEN1KMT2A
SCHEMBL6324058 0.79 NPC1 (0.44) MEN1KMT2AKDM4ENPC1RAB9A
SCHEMBL6320449 0.79 NR1H3 (0.47) MEN1KMT2AALDH1A1MAPTTP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1230210-A1 AMINOALCOHOL DERIVATIVES USEFUL FOR THE TREATMENT OF GASTROINTESTINAL DISORDERS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2002-08-14 EP disclosed
WO-2001036375-A1 AMINOALCOHOL DERIVATIVES USEFUL FOR THE TREATMENT OF GASTROINTESTINAL DISORDERS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-05-25 WO disclosed