SCHEMBL7604462

SCHEMBL7604462

O=[N+]([O-])c1cc([C@@H](O)CN(CCC(c2ccc(N3CCCC3)cc2)c2ccc(N3CCCC3)cc2)Cc2ccccc2)ccc1OCc1ccccc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.46
MAPT P10636 6/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
CTSV O60911 3/20 0.38
CTSL P07711 3/20 0.38
PDCD1 Q15116 1/20 0.37
CD274 Q9NZQ7 1/20 0.37
ALDH1A1 P00352 3/20 0.37
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
MAPK1 P28482 2/20 0.37
KDM4E B2RXH2 1/20 0.37
TP53 P04637 1/20 0.37
GAA P10253 1/20 0.37
ALOX12 P18054 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7605039 0.88 CTSV (0.42) POLBMAPTCTSVCTSLPDCD1
SCHEMBL7605286 0.86 MEN1 (0.39) MAPTALDH1A1MEN1KMT2AMAPK1
SCHEMBL7605016 0.85 MAPT (0.43) POLBMAPTNPSR1CTSVCTSL
SCHEMBL7685567 0.82 ADRB3 (0.43) MAPTALDH1A1MEN1KMT2AMAPK1
SCHEMBL7685564 0.82 ADRB3 (0.43) MAPTALDH1A1MEN1KMT2AMAPK1
SCHEMBL7607649 0.80 CTSV (0.44) POLBMAPTCTSVCTSLPDCD1
SCHEMBL7606577 0.80 CTSV (0.44) POLBMAPTCTSVCTSLPDCD1
SCHEMBL7604658 0.79 MAPT (0.44) POLBMAPTCTSVCTSLPDCD1
SCHEMBL7605323 0.79 CTSV (0.43) POLBMAPTCTSVCTSLPDCD1
SCHEMBL7611581 0.77 ALDH1A1 (0.46) POLBMAPTCYP1A2CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1230210-A1 AMINOALCOHOL DERIVATIVES USEFUL FOR THE TREATMENT OF GASTROINTESTINAL DISORDERS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2002-08-14 EP disclosed
WO-2001036375-A1 AMINOALCOHOL DERIVATIVES USEFUL FOR THE TREATMENT OF GASTROINTESTINAL DISORDERS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-05-25 WO disclosed