SCHEMBL7605972

SCHEMBL7605972

COc1ccc(C(CN(Cc2ccccc2)[C@@H](CO)c2ccc(OCc3ccccc3)c(NC(N)=O)c2)c2ccc(OC)cc2)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.44
KDM4E B2RXH2 1/20 0.44
CYP1A2 P05177 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
C5AR1 P21730 1/20 0.42
NR1H3 Q13133 2/20 0.42
MAPT P10636 3/20 0.39
EPOR P19235 1/20 0.39
F2 P00734 1/20 0.39
F10 P00742 1/20 0.39
PRSS1 P07477 1/20 0.39
PRSS2 P07478 1/20 0.39
F7 P08709 1/20 0.39
F3 P13726 1/20 0.39
PRSS3 P35030 1/20 0.39
MTNR1A P48039 1/20 0.38
MTNR1B P49286 1/20 0.38
MEN1 O00255 2/20 0.38
TP53 P04637 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7611191 0.93 ALDH1A1 (0.44) ALDH1A1KDM4ECYP1A2CYP2C9CYP2C19
SCHEMBL7606579 0.88 NR1H3 (0.43) ALDH1A1C5AR1NR1H3MAPTEPOR
SCHEMBL7606168 0.86 PTPN2 (0.41) ALDH1A1KDM4ECYP1A2CYP2C9CYP2C19
SCHEMBL7610365 0.85 AOC3 (0.40) ALDH1A1C5AR1NR1H3MAPTEPOR
SCHEMBL7611109 0.85 AOC3 (0.40) ALDH1A1C5AR1NR1H3MAPTEPOR
SCHEMBL7605952 0.83 NR1H3 (0.48) ALDH1A1KDM4ECYP1A2CYP2C9CYP2C19
SCHEMBL7606221 0.79 NPC1 (0.46) KDM4EC5AR1F2F10PRSS1
SCHEMBL7610067 0.79 AR (0.38) ALDH1A1MAPTMEN1KMT2A
SCHEMBL7608227 0.78 PTGS1 (0.40) CYP1A2CYP2C19MAPTEPORSMN1; SMN2
SCHEMBL7614703 0.78 SMN1; SMN2 (0.41) ALDH1A1KDM4EMAPTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1230210-A1 AMINOALCOHOL DERIVATIVES USEFUL FOR THE TREATMENT OF GASTROINTESTINAL DISORDERS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2002-08-14 EP disclosed
WO-2001036375-A1 AMINOALCOHOL DERIVATIVES USEFUL FOR THE TREATMENT OF GASTROINTESTINAL DISORDERS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-05-25 WO disclosed