SCHEMBL7606579

SCHEMBL7606579

COc1ccc(C(CN(Cc2ccccc2)[C@H](CO)c2ccc(OCc3ccccc3)c(C(N)=O)c2)c2ccc(OC)cc2)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1H3 Q13133 4/20 0.43
LMNA P02545 2/20 0.40
HTT P42858 2/20 0.40
ALDH1A1 P00352 2/20 0.40
MAPT P10636 2/20 0.40
C5AR1 P21730 1/20 0.40
ALOX5 P09917 1/20 0.39
LRRK2 Q5S007 1/20 0.39
TSHR P16473 2/20 0.39
MEN1 O00255 1/20 0.39
NPC1 O15118 1/20 0.39
TP53 P04637 1/20 0.39
HPGD P15428 1/20 0.39
RAB9A P51151 1/20 0.39
KMT2A Q03164 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
HDAC8 Q9BY41 1/20 0.39
EPOR P19235 1/20 0.38
TDP1 Q9NUW8 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7606168 0.91 PTPN2 (0.41) NR1H3HTTALDH1A1MAPTLRRK2
SCHEMBL7605972 0.88 ALDH1A1 (0.44) NR1H3LMNAHTTALDH1A1MAPT
SCHEMBL7611109 0.87 AOC3 (0.40) NR1H3ALDH1A1MAPTC5AR1TSHR
SCHEMBL7610365 0.87 AOC3 (0.40) NR1H3ALDH1A1MAPTC5AR1TSHR
SCHEMBL7611191 0.84 ALDH1A1 (0.44) NR1H3ALDH1A1MAPTC5AR1LRRK2
SCHEMBL7606574 0.83 NR1H3 (0.49) NR1H3LMNAHTTALDH1A1MAPT
SCHEMBL7605885 0.82 MAPT (0.45) LMNAHTTALDH1A1MAPTLRRK2
SCHEMBL7608227 0.80 PTGS1 (0.40) LMNAMAPTALOX5RAB9ASMN1; SMN2
SCHEMBL7610616 0.78 ALDH1A1 (0.43) NR1H3LMNAHTTALDH1A1MAPT
SCHEMBL4728111 0.77 KMT2A (0.43) LMNAHTTALDH1A1MAPTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1230210-A1 AMINOALCOHOL DERIVATIVES USEFUL FOR THE TREATMENT OF GASTROINTESTINAL DISORDERS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2002-08-14 EP disclosed
WO-2001036375-A1 AMINOALCOHOL DERIVATIVES USEFUL FOR THE TREATMENT OF GASTROINTESTINAL DISORDERS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-05-25 WO disclosed