SCHEMBL7605952

SCHEMBL7605952

COc1ccc(C(CN(Cc2ccccc2)C[C@H](O)c2ccc(OCc3ccccc3)c(NC(N)=O)c2)c2ccc(OC)cc2)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1H3 Q13133 6/20 0.48
ALDH1A1 P00352 3/20 0.46
KDM4E B2RXH2 1/20 0.46
CYP1A2 P05177 1/20 0.46
CYP2C9 P11712 1/20 0.46
CYP2C19 P33261 1/20 0.46
C5AR1 P21730 1/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
NPC1 O15118 1/20 0.40
POLB P06746 1/20 0.40
MAPT P10636 1/20 0.40
MMP1 P03956 1/20 0.40
MMP2 P08253 1/20 0.40
MMP9 P14780 1/20 0.40
MMP13 P45452 1/20 0.40
F2 P00734 1/20 0.39
F10 P00742 1/20 0.39
PRSS1 P07477 1/20 0.39
PRSS2 P07478 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7611188 0.93 ALDH1A1 (0.46) NR1H3ALDH1A1KDM4ECYP1A2CYP2C9
SCHEMBL7606574 0.87 NR1H3 (0.49) NR1H3ALDH1A1MEN1KMT2ANPC1
SCHEMBL7606163 0.85 NR1H3 (0.47) NR1H3ALDH1A1KDM4ECYP1A2CYP2C9
SCHEMBL7610361 0.85 NR1H3 (0.46) NR1H3ALDH1A1KDM4ECYP1A2CYP2C9
SCHEMBL7611102 0.85 NR1H3 (0.46) NR1H3ALDH1A1KDM4ECYP1A2CYP2C9
SCHEMBL7605972 0.83 ALDH1A1 (0.44) NR1H3ALDH1A1KDM4ECYP1A2CYP2C9
SCHEMBL7606219 0.79 NPC1 (0.47) NR1H3KDM4EC5AR1MEN1KMT2A
SCHEMBL7610085 0.78 HDAC3 (0.44) NR1H3ALDH1A1KDM4ECYP1A2CYP2C9
SCHEMBL7608224 0.78 MMP1 (0.45) NR1H3CYP1A2CYP2C19MAPTMMP1
SCHEMBL7695645 0.78 MMP1 (0.45) NR1H3CYP1A2CYP2C19MAPTMMP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1230210-A1 AMINOALCOHOL DERIVATIVES USEFUL FOR THE TREATMENT OF GASTROINTESTINAL DISORDERS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2002-08-14 EP disclosed
WO-2001036375-A1 AMINOALCOHOL DERIVATIVES USEFUL FOR THE TREATMENT OF GASTROINTESTINAL DISORDERS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-05-25 WO disclosed