SCHEMBL760652

SCHEMBL760652

O=C(O)c1coc2c1C(=O)CCC2

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 1/20 0.42
ALDH1A1 P00352 5/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
PTK2 Q05397 1/20 0.36
POLB P06746 4/20 0.35
APOBEC3A P31941 1/20 0.35
APOBEC3G Q9HC16 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
HPGD P15428 3/20 0.35
MAOB P27338 1/20 0.34
KDM4E B2RXH2 3/20 0.33
RORC P51449 1/20 0.33
RXFP1 Q9HBX9 1/20 0.33
LDHA P00338 1/20 0.32
NTRK3 Q16288 1/20 0.32
NTRK2 Q16620 1/20 0.32
HSD17B10 Q99714 2/20 0.32
MAPT P10636 1/20 0.32
GAA P10253 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6762871 0.96 NAMPT (0.40) NAMPTALDH1A1SMN1; SMN2PTK2POLB
SCHEMBL6948898 0.89 MAOB (0.36) NAMPTMAOBLDHANTRK3NTRK2
SCHEMBL5189062 0.84 NAMPT (0.41) NAMPTALDH1A1SMN1; SMN2HPGDKDM4E
SCHEMBL5444456 0.84 NAMPT (0.41) NAMPTALDH1A1SMN1; SMN2POLBHPGD
SCHEMBL5236831 0.80 L3MBTL1 (0.42) NAMPTALDH1A1SMN1; SMN2POLBTDP1
SCHEMBL5233483 0.78 POLB (0.48) SMN1; SMN2POLBMAPT
SCHEMBL5233488 0.78 POLB (0.48) SMN1; SMN2POLBMAPT
SCHEMBL5238254 0.78 POLB (0.48) SMN1; SMN2POLBMAPT
SCHEMBL16931551 0.77 CDK5 (0.36) NAMPTALDH1A1PTK2L3MBTL1HPGD
SCHEMBL4899883 0.77 BRD4 (0.47) ALDH1A1SMN1; SMN2HPGDMAOBKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 139 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1754705-A2 Antagonists for treatment of CD11/CD18 adhesion receptor mediated disorders Genentech, Inc. (US) 2007-02-21 EP claimed
US-6936620-B2 Barbituric acid derivatives as inhibitors of TNF-α converting enzyme (TACE) and/or matrix metalloproteinases BRISTOL MYERS SQUIBB COMPANY (US) 2005-08-30 US claimed
US-6599918-B2 Inhibit Factor Xa Factor IIa (thrombin) AVENTIS PHARMACEUTICALS INC. 2003-07-29 US claimed
US-20020193410-A1 Substituted (aminoiminomethyl or aminomethyl) dihydrobenzofurans and benzopyrans AVENTIS PHARMACEUTICALS INC. 2002-12-19 US claimed
EP-3710428-B1 MODULATORS OF THE INTEGRATED STRESS PATHWAY CALICO LIFE SCIENCES LLC (US) 2026-03-25 EP disclosed
CN-121045114-A Compound TBFC-I and preparation method and application thereof 农业农村部规划设计研究院 2025-12-02 CN disclosed
US-20240392220-A1 BRANDY REPLICAS AVA FOOD LABS, INC. 2024-11-28 US disclosed
US-20240307382-A1 MODULATORS OF THE INTEGRATED STRESS PATHWAY ABBVIE INC. 2024-09-19 US disclosed
EP-4408967-A1 BRANDY REPLICAS AVA FOOD LABS, INC. (US) 2024-08-07 EP disclosed
CN-118339274-A Brandy replica 艾娃食品实验室股份有限公司 2024-07-12 CN disclosed
CN-112204009-B Modulators of integrated stress pathways 卡里科生命科学有限责任公司 2024-05-07 CN disclosed
CN-115943957-B Application of TBFC in preparation of medicines for preventing and treating bacterial diseases 北京景霁智惠科技有限公司 2024-01-26 CN disclosed
EP-0725775-A1 CERTAIN FUSED PYRROLECARBOXANILIDES; A NEW CLASS OF GABA BRAIN RECEPTOR LIGANDS NEUROGEN CORPORATION (US) 1996-08-14 EP disclosed
WO-1996022294-A1 BICYCLIC BENZAZEPINE DERIVATIVES AS VASOPRESSIN ANTAGONISTS AMERICAN CYANAMID COMPANY (US) 1996-07-25 WO disclosed
WO-1996022295-A1 TRICYCLIC BENZAZEPINE VASOPRESSIN ANTAGONISTS AMERICAN CYANAMID COMPANY (US) 1996-07-25 WO disclosed
US-5532235-A TO TREAT EXCESS RENAL REABSORPTION AMERICAN CYANAMID COMPANY (US) 1996-07-02 US disclosed
US-5484944-A ANXIETY, SLEEP, MEMORY NEUROGEN CORPORATION (US) 1996-01-16 US disclosed
WO-1995011885-A1 CERTAIN FUSED PYRROLECARBOXANILIDES; A NEW CLASS OF GABA BRAIN RECEPTOR LIGANDS NEUROGEN CORPORATION (US) 1995-05-04 WO disclosed
US-4336202-A 1,3-Cyclohexanedione derivatives KURARAY CO., LTD. (JP) 1982-06-22 US disclosed
EP-0041656-A2 Cyclohexanone derivatives and preparation thereof KURARAY CO., LTD. (JP) 1981-12-16 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240307382-A1 MODULATORS OF THE INTEGRATED STRESS PATHWAY ATF4, ATF1, DDIT3 NAMPT 2047/4885ALDH1A1 3433/4885SMN1; SMN2 2486/4885
US-20020193410-A1 Substituted (aminoiminomethyl or aminomethyl) dihydrobenzofurans and benzopyrans F2, TFPI, F3 NAMPT 2067/4885ALDH1A1 1396/4885SMN1; SMN2 2200/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.