SCHEMBL7606604

SCHEMBL7606604

COc1ccc(C(CCN(Cc2ccccc2)[C@H](CO)c2ccc(OCc3ccccc3)c(CO)c2)c2ccc(OC)cc2)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.43
MAPT P10636 2/20 0.43
MEN1 O00255 3/20 0.42
KMT2A Q03164 3/20 0.42
NPC1 O15118 1/20 0.42
LMNA P02545 1/20 0.42
TP53 P04637 1/20 0.42
HPGD P15428 1/20 0.42
HTT P42858 1/20 0.42
RAB9A P51151 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
ABCB1 P08183 3/20 0.41
ELANE P08246 1/20 0.39
CTSG P08311 1/20 0.39
SLC1A5 Q15758 1/20 0.39
C5AR1 P21730 1/20 0.39
MTNR1A P48039 2/20 0.39
MTNR1B P49286 2/20 0.39
HTR1A P08908 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7610616 0.89 ALDH1A1 (0.43) ALDH1A1MAPTMEN1KMT2ANPC1
SCHEMBL7605885 0.85 MAPT (0.45) ALDH1A1MAPTMEN1KMT2ANPC1
SCHEMBL7605019 0.85 MAPT (0.43) ALDH1A1MAPTMEN1KMT2ANPC1
SCHEMBL7606596 0.82 NR1H3 (0.43) ALDH1A1MAPTMEN1KMT2ANPC1
SCHEMBL7610096 0.82 HDAC3 (0.44) ALDH1A1MAPTMEN1KMT2ANPC1
SCHEMBL7608457 0.82 BCHE (0.41) MAPTLMNARAB9ASMN1; SMN2BCHE
SCHEMBL7610365 0.79 AOC3 (0.40) ALDH1A1MAPTNPC1RAB9ANPSR1
SCHEMBL7611109 0.79 AOC3 (0.40) ALDH1A1MAPTNPC1RAB9ANPSR1
SCHEMBL7614716 0.77 ALOX5 (0.39) BCHE
SCHEMBL7606168 0.76 PTPN2 (0.41) ALDH1A1MAPTNPC1HTTRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1230210-A1 AMINOALCOHOL DERIVATIVES USEFUL FOR THE TREATMENT OF GASTROINTESTINAL DISORDERS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2002-08-14 EP disclosed
WO-2001036375-A1 AMINOALCOHOL DERIVATIVES USEFUL FOR THE TREATMENT OF GASTROINTESTINAL DISORDERS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-05-25 WO disclosed